SCHEMBL9769346

SCHEMBL9769346

C=Cc1cnc(NC(=O)C(C)C)nc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 2/20 0.41
CCNE1 P24864 1/20 0.41
CDK2 P24941 1/20 0.41
TSHR P16473 2/20 0.40
ADORA1 P30542 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
RECQL P46063 1/20 0.39
ALDH1A1 P00352 3/20 0.37
LMNA P02545 3/20 0.37
HSD17B10 Q99714 1/20 0.37
MAPK1 P28482 1/20 0.37
NPC1 O15118 1/20 0.37
TP53 P04637 1/20 0.37
RAB9A P51151 1/20 0.37
HTT P42858 2/20 0.36
NOS1 P29475 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CDK5R1 Q15078 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9769174 0.79 ALDH1A1 (0.49) CDK5CCNE1CDK2TSHRSMN1; SMN2
SCHEMBL9769380 0.77 CCNE1 (0.45) CDK5CCNE1CDK2TSHRADORA1
SCHEMBL9769158 0.76 CCNE1 (0.39) CDK5CCNE1CDK2TSHRADORA1
SCHEMBL10584279 0.75 LMNA (0.53) CDK5CCNE1CDK2TSHRADORA1
SCHEMBL9769375 0.73 CCNE1 (0.40) CDK5CCNE1CDK2TSHRADORA1
SCHEMBL19699602 0.72 TSHR (0.39) CDK5CCNE1CDK2TSHRADORA1
SCHEMBL20819348 0.72 ALDH1A1 (0.39) CDK5CCNE1CDK2TSHRADORA1
SCHEMBL19699611 0.72 TSHR (0.39) CDK5CCNE1CDK2TSHRADORA1
SCHEMBL9769330 0.71 ADRB2 (0.44) TSHRSMN1; SMN2LMNAMEN1KMT2A
SCHEMBL1447828 0.71 TSHR (0.44) CDK5CCNE1CDK2TSHRADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5019578-A β-adrenergic agonists MERCK & CO., INC. (US) 1991-05-28 US disclosed
EP-0318092-A2 Novel beta-adrenergic agonists MERCK & CO. INC. (US) 1989-05-31 EP disclosed
US-4816457-A HYPOTENSIVE AGENTS, BRONCHODILATORS, EYES MERCK & CO., INC., A CORP. OF NJ 1989-03-28 US disclosed