SCHEMBL9769158

SCHEMBL9769158

CC(C)C(=O)Nc1ncc(C(O)CBr)cn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNE1 P24864 1/20 0.39
CDK2 P24941 1/20 0.39
CDK5 Q00535 1/20 0.39
MAPK1 P28482 1/20 0.38
TSHR P16473 2/20 0.37
ADORA1 P30542 1/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
RECQL P46063 1/20 0.36
P2RX3 P56373 1/20 0.36
P2RX2 Q9UBL9 1/20 0.36
FFAR2 O15552 1/20 0.35
ALDH1A1 P00352 3/20 0.35
LMNA P02545 2/20 0.35
HSD17B10 Q99714 1/20 0.35
RAB9A P51151 2/20 0.35
NPC1 O15118 1/20 0.35
TP53 P04637 1/20 0.35
POLB P06746 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10588784 0.84 LMNA (0.35) CCNE1CDK2ADORA1ALDH1A1LMNA
SCHEMBL9769330 0.80 ADRB2 (0.44) TSHRSMN1; SMN2LMNAMEN1KMT2A
SCHEMBL28891535 0.79 P2RX3 (0.37) CCNE1CDK2CDK5MAPK1TSHR
SCHEMBL20819399 0.76 SMN1; SMN2 (0.40) SMN1; SMN2RECQLFFAR2ALDH1A1HTT
SCHEMBL20832742 0.76 SMN1; SMN2 (0.40) SMN1; SMN2RECQLFFAR2ALDH1A1HTT
SCHEMBL9769380 0.76 CCNE1 (0.45) CCNE1CDK2CDK5TSHRADORA1
SCHEMBL9769375 0.76 CCNE1 (0.40) CCNE1CDK2CDK5MAPK1TSHR
SCHEMBL9769346 0.76 CDK5 (0.41) CCNE1CDK2CDK5MAPK1TSHR
Hydrochloric Acid SCHEMBL20819391 0.76 SMN1; SMN2 (0.39) SMN1; SMN2RECQLALDH1A1
Hydrochloric Acid SCHEMBL20819389 0.76 SMN1; SMN2 (0.39) SMN1; SMN2RECQLALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5019578-A β-adrenergic agonists MERCK & CO., INC. (US) 1991-05-28 US disclosed
EP-0318092-A2 Novel beta-adrenergic agonists MERCK & CO. INC. (US) 1989-05-31 EP disclosed
US-4816457-A HYPOTENSIVE AGENTS, BRONCHODILATORS, EYES MERCK & CO., INC., A CORP. OF NJ 1989-03-28 US disclosed