SCHEMBL977331

SCHEMBL977331

O=S(=O)(OCC(F)(F)C(F)F)C(F)(F)F

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.34
CA1 P00915 2/20 0.33
CA9 Q16790 1/20 0.33
POLB P06746 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
ALDH1A1 P00352 2/20 0.32
TP53 P04637 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2488623 0.83 CA2 (0.33) CA2CA1CA9
SCHEMBL17491120 0.81 CA1 (0.41) CA2CA1CA9POLBTDP1
SCHEMBL76110 0.78 CA2 (0.42) CA2CA1
SCHEMBL19348714 0.77 CA1 (0.60) CA2CA1CA9MEN1KMT2A
SCHEMBL1979109 0.77 ALDH1A1 (0.37) CA2CA1CA9POLBMEN1
SCHEMBL17466437 0.77 CA1 (0.33) CA2CA1CA9POLBTDP1
SCHEMBL7257180 0.77 ALDH1A1 (0.35) CA2CA1CA9POLBMEN1
SCHEMBL17456472 0.76 MEN1 (0.35) CA2CA1CA9MEN1KMT2A
SCHEMBL17456443 0.76 CA1 (0.32) CA2CA1CA9POLBTDP1
SCHEMBL17456469 0.76 CA1 (0.32) CA2CA1CA9POLBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 274 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10633357-B2 Intermediates and process for preparing intermediates in the production of substituted pyrazolopyridines ADVERIO PHARMA GMBH (DE) 2020-04-28 US claimed
US-20190177288-A1 INTERMEDIATES AND PROCESS FOR PREPARING INTERMEDIATES IN THE PRODUCTION OF SUBSTITUTED PYRAZOLOPYRIDINES ADVERIO PHARMA GMBH (DE) 2019-06-13 US claimed
US-20180065942-A1 CRYSTALLINE SUBSTITUTED 5-FLUORO-1H-PYRAZOLOPYRIDINES AND PROCESS FOR PREPARING ADVERIO PHARMA GMBH (DE) 2018-03-08 US claimed
US-9845300-B2 Process for preparing substituted 5-fluoro-1H-pyrazolopyridines ADVERIO PHARMA GMBH (DE) 2017-12-19 US claimed
US-20170158652-A1 PROCESS FOR PREPARING SUBSTITUTED 5-FLUORO-1H-PYRAZOLOPYRIDINES ADVERIO PHARMA GMBH (DE) 2017-06-08 US claimed
EP-2896617-B1 METHOD FOR PRODUCING SUBSTITUTED (Z)-ALPHA-FLUORO-BETA-AMINO-ACRYLALDEHYDES ADVERIO PHARMA GMBH (DE) 2016-10-05 EP claimed
US-20160009671-A1 PROCESS FOR PREPARING SUBSTITUTED 5-FLUORO-1H-PYRAZOLOPYRIDINES ADVERIO PHARMA GMBH (DE) 2016-01-14 US claimed
EP-2896617-A1 Method for producing substituted 5-fluoro-1h-pyrazolopyridines Adverio Pharma GmbH (DE) 2015-07-22 EP claimed
US-20140315926-A1 Process for preparing substituted 5-fluoro-1H-pyrazolopyridines ADVERIO PHARMA GMBH (DE) 2014-10-23 US claimed
EP-2782914-A1 METHOD FOR PRODUCING SUBSTITUTED 5-FLUORO-1H-PYRAZOLOPYRIDINES Bayer Pharma Aktiengesellschaft (DE) 2014-10-01 EP claimed
US-20130143900-A1 Process for preparing substituted 5-fluoro-1H-pyrazolopyridines BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-06-06 US claimed
WO-2013076168-A1 METHOD FOR PRODUCING SUBSTITUTED 5-FLUORO-1H-PYRAZOLOPYRIDINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2013-05-30 WO claimed
EP-4739675-A1 INDOLE DERIVATIVES WITH FACTOR B INHIBITORY ACTIVITY Sitala Bio Ltd (GB) 2026-05-13 EP disclosed
EP-4739667-A2 INDOLE DERIVATIVES WITH FACTOR B INHIBITORY ACTIVITY Sitala Bio Ltd (GB) 2026-05-13 EP disclosed
EP-3976604-B1 1,3,4-OXADIAZOLE DERIVATIVE COMPOUNDS AS HISTONE DEACETYLASE 6 INHIBITOR, AND THE PHARMACEUTICAL COMPOSITION COMPRISING THE SAME CHONG KUN DANG PHARMACEUTICAL CORP (KR) 2026-01-21 EP disclosed
US-12440484-B2 1,3,4-oxadiazole homophthalimide derivative compounds as histone deacetylase 6 inhibitor, and the pharmaceutical composition comprising the same CHONG KUN DANG PHARMACEUTICAL CORPORATION (KR) 2025-10-14 US disclosed
US-20050009838-A1 Piperidinyl-and piperazinyl-sulfonylmethyl hydroxamic acids and their use as protease inhibitors PHARMACIA CORPORATION 2005-01-13 US disclosed
US-20040138065-A1 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2004-07-15 US disclosed
EP-1385817-A2 MALONONITRILE COMPOUNDS AND THEIR USE AS PESTICIDES SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2004-02-04 EP disclosed
WO-2002090320-A2 MALONONITRILE COMPOUNDS AND THEIR USE AS PESTICIDES SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2002-11-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170158652-A1 PROCESS FOR PREPARING SUBSTITUTED 5-FLUORO-1H-PYRAZOLOPYRIDINES CYP3A5, CYP4F2, CYP2F1 CA2 3178/4885CA1 4728/4885CA9 3916/4885
US-20180065942-A1 CRYSTALLINE SUBSTITUTED 5-FLUORO-1H-PYRAZOLOPYRIDINES AND PROCESS FOR PREPARING CYP3A5, CYP2F1, CYP4F2 CA2 1874/4885CA1 4077/4885CA9 3228/4885
US-20160009671-A1 PROCESS FOR PREPARING SUBSTITUTED 5-FLUORO-1H-PYRAZOLOPYRIDINES CYP3A5, CYP4F2, CYP2F1 CA2 3178/4885CA1 4728/4885CA9 3916/4885
US-12440484-B2 1,3,4-oxadiazole homophthalimide derivative compounds as histone deacetylase 6 inhibitor, and the pharmaceutical composition comprising the same HDAC1, HDAC11, HDAC3 CA2 1703/4885CA1 1969/4885CA9 1509/4885
US-20040138065-A1 Malononitrile compounds and their use as pesticides CBR1, MAL2, CBR3 CA2 118/4885CA1 754/4885CA9 404/4885
US-20050009838-A1 Piperidinyl-and piperazinyl-sulfonylmethyl hydroxamic acids and their use as protease inhibitors MMP1, PREP, MMP3 CA2 101/4885CA1 79/4885CA9 147/4885
US-10633357-B2 Intermediates and process for preparing intermediates in the production of substituted pyrazolopyridines CYP3A5, CYP4F2, CYP2F1 CA2 2527/4885CA1 4462/4885CA9 3623/4885
US-20130143900-A1 Process for preparing substituted 5-fluoro-1H-pyrazolopyridines CYP3A5, CYP4F2, CYP2F1 CA2 3178/4885CA1 4728/4885CA9 3916/4885
US-20140315926-A1 Process for preparing substituted 5-fluoro-1H-pyrazolopyridines CYP3A5, CYP4F2, CYP2F1 CA2 3178/4885CA1 4728/4885CA9 3916/4885
US-20190177288-A1 INTERMEDIATES AND PROCESS FOR PREPARING INTERMEDIATES IN THE PRODUCTION OF SUBSTITUTED PYRAZOLOPYRIDINES CYP3A5, CYP4F2, CYP2F1 CA2 2527/4885CA1 4462/4885CA9 3623/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.