SCHEMBL9775920

SCHEMBL9775920

COn1cc(C(=O)O)c(=O)c2cc3cc(F)c(N4CCN(C)CC4)cc3nc21

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.52
DRD3 P35462 1/20 0.52
LMNA P02545 3/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
KDM4E B2RXH2 13/20 0.48
HPGD P15428 7/20 0.48
NPC1 O15118 1/20 0.48
HSD17B10 Q99714 6/20 0.41
ADRA2B P18089 1/20 0.41
MAPK1 P28482 1/20 0.41
GAA P10253 1/20 0.41
RAD52 P43351 1/20 0.41
MAPT P10636 1/20 0.40
BRD4 O60885 1/20 0.40
TSHR P16473 1/20 0.40
HTT P42858 1/20 0.40
CYP2J2 P51589 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
ALB P02768 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9775973 0.90 ALDH1A1 (0.52) ALDH1A1DRD3LMNAMEN1KMT2A
SCHEMBL9775869 0.88 KDM4E (0.47) ALDH1A1DRD3MEN1KMT2AKDM4E
SCHEMBL9094359 0.88 ALDH1A1 (0.55) ALDH1A1DRD3LMNAMEN1KMT2A
Hydrochloric Acid SCHEMBL9097124 0.87 ALDH1A1 (0.54) ALDH1A1DRD3LMNAMEN1KMT2A
SCHEMBL8941977 0.85 KMT2A (0.38) ALDH1A1DRD3LMNAMEN1KMT2A
SCHEMBL9775890 0.85 DRD3 (0.67) ALDH1A1DRD3LMNAMEN1KMT2A
SCHEMBL9775907 0.85 ALDH1A1 (0.52) ALDH1A1DRD3LMNAMEN1KMT2A
SCHEMBL9775969 0.85 ALDH1A1 (0.67) ALDH1A1DRD3LMNAMEN1KMT2A
SCHEMBL8942417 0.84 LMNA (0.39) ALDH1A1LMNAMEN1KMT2AKDM4E
SCHEMBL8942065 0.84 TOP1 (0.41) ALDH1A1LMNAKMT2AKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5004745-A Benzo[1,8]naphthyridine derivatives, their preparation and the compositions which contain them LABORATOIRE ROGER BELLON (FR) 1991-04-02 US disclosed
US-4990515-A Chemical intermediates RHONE-POULENC SANTE (FR) 1991-02-05 US disclosed
US-4970213-A Benzo(1,8)naphthyridine derivatives as intermediates RHONE-POULENC SANTE (FR) 1990-11-13 US disclosed