SCHEMBL8942417

SCHEMBL8942417

COn1cc(C(=O)O)c(=O)c2cc3cc(F)c(F)cc3nc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.39
CYP2C9 P11712 1/20 0.39
ATP6V1B2 P21281 1/20 0.39
TBXA2R P21731 1/20 0.39
EDNRA P25101 1/20 0.39
TARBP2 Q15633 1/20 0.39
TOP2A P11388 3/20 0.37
TOP2B Q02880 3/20 0.37
DPP4 P27487 4/20 0.35
CHRM2 P08172 1/20 0.35
DRD1 P21728 1/20 0.35
KMT2A Q03164 2/20 0.35
ABCC4 O15439 2/20 0.35
MEN1 O00255 1/20 0.35
PKM P14618 1/20 0.35
PTGS1 P23219 1/20 0.35
GSK3B P49841 3/20 0.34
EPHA2 P29317 1/20 0.34
FLT4 P35916 1/20 0.34
RARB P10826 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9536515 0.88 LMNA (0.32) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL9775901 0.86 TOP2A (0.38) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL8942074 0.85 KMT2A (0.46) LMNAKMT2AMEN1KDM4EHSD17B10
SCHEMBL9775920 0.84 ALDH1A1 (0.52) LMNAKMT2AMEN1KDM4EHSD17B10
SCHEMBL9775973 0.84 ALDH1A1 (0.52) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL6605949 0.84 LMNA (0.41) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL8942372 0.83 TOP2A (0.33) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL8941977 0.83 KMT2A (0.38) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL8942065 0.82 TOP1 (0.41) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL8942028 0.81 LMNA (0.59) LMNACYP2C9ATP6V1B2TBXA2REDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0379413-B1 1,8-Benzonaphthyridine derivatives, their production and compositions containing them BELLON LABOR SA ROGER (FR) 1993-12-22 EP claimed
US-4990515-A Chemical intermediates RHONE-POULENC SANTE (FR) 1991-02-05 US claimed
US-5556861-A 1,8 benzonaphthyridine derivatives and antimicrobial compositions LABORATOIRE ROGER BELLON (FR) 1996-09-17 US disclosed
US-5053509-A Microbiocides; AIDS LABORATOIRE ROGER BELLON (FR) 1991-10-01 US disclosed
US-5004745-A Benzo[1,8]naphthyridine derivatives, their preparation and the compositions which contain them LABORATOIRE ROGER BELLON (FR) 1991-04-02 US disclosed
US-4990515-A Chemical intermediates RHONE-POULENC SANTE (FR) 1991-02-05 US disclosed
US-4970213-A Benzo(1,8)naphthyridine derivatives as intermediates RHONE-POULENC SANTE (FR) 1990-11-13 US disclosed