SCHEMBL9780222

SCHEMBL9780222

C[C@@H](CC(=O)O)C(=O)c1ccc(C(=S)N(C)C)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.47
MAPT P10636 4/20 0.47
HDAC3 O15379 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC10 Q969S8 1/20 0.45
HDAC11 Q96DB2 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
HDAC9 Q9UKV0 1/20 0.45
HDAC5 Q9UQL6 1/20 0.45
HSP90AA1 P07900 2/20 0.37
HSP90AB1 P08238 1/20 0.37
MMP2 P08253 2/20 0.36
MMP9 P14780 2/20 0.36
MMP12 P39900 2/20 0.36
MMP14 P50281 1/20 0.36
MMP15 P51511 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10911181 1.00 ALDH1A1 (0.47) ALDH1A1MAPTHDAC3HDAC4HDAC1
SCHEMBL10353455 0.84 HDAC3 (0.49) ALDH1A1MAPTHDAC3HDAC4HDAC1
SCHEMBL9780324 0.83 ALDH1A1 (0.40) ALDH1A1MAPTHDAC3HDAC4HDAC1
SCHEMBL8775491 0.78 CHRM2 (0.53) ALDH1A1MAPTHDAC3HDAC4HDAC1
SCHEMBL7325551 0.78 LMNA (0.53) MAPTHDAC3HDAC4HDAC1HDAC7
SCHEMBL9780294 0.77 ALDH1A1 (0.43) ALDH1A1MAPTHSP90AA1HSP90AB1HSD17B10
SCHEMBL9780297 0.77 ALDH1A1 (0.43) ALDH1A1MAPTHSP90AA1HSP90AB1HSD17B10
SCHEMBL8823315 0.77 PGR (0.52) ALDH1A1MAPTMMP2MMP9MMP12
SCHEMBL135357 0.77 PGR (0.52) ALDH1A1MAPTMMP2MMP9MMP12
SCHEMBL8381806 0.76 MAPT (0.44) ALDH1A1MAPTHDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0206741-B1 LEUKOTRIENE ANTAGONISTS MERCK FROSST CANADA INC. (CA) 1991-04-10 EP disclosed
US-4990526-A Skin disorders, antiallergens, antiinflammatory agents MERCK FROSST CANADA, INC. (CA) 1991-02-05 US disclosed
EP-0206741-A2 Leukotriene antagonists MERCK FROSST CANADA INC. (CA) 1986-12-30 EP disclosed