SCHEMBL9780294

SCHEMBL9780294

CC(CC(=O)O)[C@H](O)c1ccc(C(=S)N(C)C)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
MAPT P10636 1/20 0.43
GAA P10253 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
USP5 P45974 1/20 0.36
CYSLTR2 Q9NS75 1/20 0.35
CYSLTR1 Q9Y271 1/20 0.35
HSP90AA1 P07900 1/20 0.35
HSP90AB1 P08238 1/20 0.35
FFAR1 O14842 3/20 0.34
KDM4E B2RXH2 1/20 0.33
CYP2C9 P11712 1/20 0.33
HPGD P15428 1/20 0.33
CYP2C19 P33261 1/20 0.33
BACE1 P56817 1/20 0.33
HSD17B10 Q99714 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9780297 1.00 ALDH1A1 (0.43) ALDH1A1MAPTGAAL3MBTL1USP5
SCHEMBL10911181 0.77 ALDH1A1 (0.47) ALDH1A1MAPTGAAL3MBTL1HSP90AA1
SCHEMBL9780222 0.77 ALDH1A1 (0.47) ALDH1A1MAPTGAAL3MBTL1HSP90AA1
SCHEMBL9734675 0.75 CYSLTR2 (0.41) ALDH1A1GAAL3MBTL1CYSLTR2CYSLTR1
SCHEMBL9863050 0.75 CYSLTR2 (0.36) ALDH1A1GAAL3MBTL1USP5CYSLTR2
SCHEMBL9780346 0.74 FFAR1 (0.39) ALDH1A1GAAL3MBTL1USP5CYSLTR2
SCHEMBL9732958 0.66 POLB (0.51) ALDH1A1GAAL3MBTL1CYSLTR2CYSLTR1
SCHEMBL11823552 0.66 MME (0.47) FFAR1
SCHEMBL10547785 0.65 CYSLTR2 (0.53) ALDH1A1L3MBTL1CYSLTR2CYSLTR1FFAR1
SCHEMBL11443491 0.64 ALDH1A1 (0.50) ALDH1A1MAPTCYP2C9HPGDCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0206741-B1 LEUKOTRIENE ANTAGONISTS MERCK FROSST CANADA INC. (CA) 1991-04-10 EP disclosed
US-4990526-A Skin disorders, antiallergens, antiinflammatory agents MERCK FROSST CANADA, INC. (CA) 1991-02-05 US disclosed
EP-0206741-A2 Leukotriene antagonists MERCK FROSST CANADA INC. (CA) 1986-12-30 EP disclosed