SCHEMBL9780236

SCHEMBL9780236

COC(=O)CC(C)C(=O)c1ccc(SCOC(=O)C(F)(F)F)cc1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.36
NPC1 O15118 2/20 0.36
TAS1R3 Q7RTX0 1/20 0.36
TAS1R1 Q7RTX1 1/20 0.36
MLYCD O95822 2/20 0.33
GAA P10253 2/20 0.31
KDM4E B2RXH2 1/20 0.31
CYP1A2 P05177 1/20 0.31
GLA P06280 1/20 0.31
CYP3A4 P08684 1/20 0.31
MAPT P10636 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
TP53 P04637 1/20 0.30
ESRRB O95718 1/20 0.30
KCNA5 P22460 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9735344 0.76 PLK1 (0.45) TAS1R3TAS1R1GAAKDM4EMAPT
SCHEMBL9734549 0.72 CA1 (0.48) CYP1A2CYP3A4ESRRBKCNA5
SCHEMBL9733852 0.71 ALDH1A1 (0.37) RAB9ATAS1R3TAS1R1GAAMAPT
SCHEMBL9780181 0.70 KCNA5 (0.38) RAB9AGAACYP1A2MAPTESRRB
SCHEMBL9733728 0.70 ALDH1A1 (0.51) CYP1A2
SCHEMBL3663713 0.70 FFAR1 (0.46) RAB9ANPC1CYP1A2CYP3A4CYP2C19
SCHEMBL8535929 0.70 KCNA5 (0.49) MAPTESRRBKCNA5
SCHEMBL9057225 0.67 HSD17B10 (0.50) GAAKDM4ECYP1A2MAPTTP53
SCHEMBL9734951 0.67 HSP90AA1 (0.35) RAB9ANPC1MLYCDMAPT
SCHEMBL9780250 0.66 KCNA5 (0.35) RAB9AGAACYP1A2MAPTESRRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4990526-A Skin disorders, antiallergens, antiinflammatory agents MERCK FROSST CANADA, INC. (CA) 1991-02-05 US disclosed
EP-0206741-A2 Leukotriene antagonists MERCK FROSST CANADA INC. (CA) 1986-12-30 EP disclosed