SCHEMBL9780857

SCHEMBL9780857

O=C(O)CCCCCOc1c(Cl)cccc1Cl

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.61
PYGL P06737 1/20 0.56
LTB4R Q15722 4/20 0.49
PPARA Q07869 3/20 0.47
MAPT P10636 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
HDAC9 Q9UKV0 1/20 0.44
HDAC5 Q9UQL6 1/20 0.44
ALDH1A1 P00352 1/20 0.44
SERPINE1 P05121 1/20 0.44
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9780778 0.98 KMT2A (0.62) KMT2APYGLLTB4RPPARASERPINE1
SCHEMBL9780586 0.93 KMT2A (0.65) KMT2APYGLHPGDL3MBTL1AKR1B1
SCHEMBL27634252 0.89 KMT2A (0.49) KMT2APYGLLTB4RPPARAMAPT
SCHEMBL9780958 0.87 KMT2A (0.67) KMT2APYGLL3MBTL1AKR1B1
SCHEMBL27654735 0.84 MAPT (0.45) KMT2APYGLLTB4RMAPTALDH1A1
SCHEMBL9501831 0.82 POLB (0.56) KMT2AMAPTHPGDL3MBTL1
SCHEMBL9322243 0.81 MEN1 (0.55) KMT2APYGLLTB4RPPARAMAPT
SCHEMBL6575170 0.80 PYGL (0.51) PYGLLTB4RALDH1A1ALB
SCHEMBL20678420 0.79 LTB4R (0.48) PYGLLTB4RPPARAMAPTRXFP1
SCHEMBL3168428 0.79 MEN1 (0.57) KMT2ALTB4RPPARAMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0257378-B1 PYRIMIDINE DERIVATIVES, THEIR PREPARATION AND MEDICAMENTS CONTAINING THESE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1991-07-03 EP disclosed
US-5010060-A Method of treating herpes simplex viral infection employing pyrimidine derivatives HOFFMANN-LA ROCHE INC. (US) 1991-04-23 US disclosed
US-4851519-A AMIDO NUCLEOSIDES, VIRICIDES HOFFMANN-LA ROCHE INC. (US) 1989-07-25 US disclosed
EP-0257378-A1 Pyrimidine derivatives, their preparation and medicaments containing these derivatives F. HOFFMANN-LA ROCHE AG (CH) 1988-03-02 EP disclosed