SCHEMBL9785451

SCHEMBL9785451

CCOC(=O)C(=C(C)C)c1cnc(C(C)(C)C)nc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FOS P01100 1/20 0.38
JUN P05412 1/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
GLO1 Q04760 1/20 0.35
ALDH1A1 P00352 5/20 0.33
MAPT P10636 2/20 0.33
KDM4E B2RXH2 2/20 0.33
PKM P14618 1/20 0.33
DGAT1 O75907 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
PRNP P04156 1/20 0.32
RAB9A P51151 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
HPGD P15428 2/20 0.32
GAA P10253 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9785366 0.83 FOS (0.40) FOSJUNNFKB1NFKB2RELA
SCHEMBL3564942 0.79 CYP2C9 (0.47) FOSJUNNFKB1NFKB2RELA
SCHEMBL10654101 0.78 TDP1 (0.33) ALDH1A1PKMKMT2A
SCHEMBL9785488 0.77 KDM4E (0.32) ALDH1A1KDM4E
SCHEMBL29117925 0.70 ALDH1A1 (0.57) ALDH1A1MAPTKDM4ERAB9AHPGD
SCHEMBL9785541 0.70 SMN1; SMN2 (0.45) FOSJUNNFKB1NFKB2RELA
SCHEMBL31292519 0.69 CNR2 (0.38) FOSJUNNFKB1NFKB2RELA
SCHEMBL8950028 0.68 SMN1; SMN2 (0.51) ALDH1A1MAPTHPGDGAAMEN1
SCHEMBL10414576 0.68 CA12 (0.54) MAPTRAB9ANPC1
SCHEMBL10414574 0.68 CA12 (0.54) MAPTRAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5010200-A Insecticide intermediates IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-04-23 US disclosed
US-4962109-A MITICIDES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-10-09 US disclosed
EP-0295839-A2 Pyrimidine derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-12-21 EP disclosed