SCHEMBL9785366

SCHEMBL9785366

CCOC(=O)C(=O)c1cnc(C(C)(C)C)nc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FOS P01100 1/20 0.40
JUN P05412 1/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
ALDH1A1 P00352 4/20 0.38
MAPT P10636 2/20 0.38
PKM P14618 1/20 0.36
KDM4E B2RXH2 2/20 0.35
DGAT1 O75907 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
RAB9A P51151 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
PRNP P04156 1/20 0.34
HPGD P15428 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
GAA P10253 1/20 0.33
NPC1 O15118 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3564942 0.83 CYP2C9 (0.47) FOSJUNNFKB1NFKB2RELA
SCHEMBL9785451 0.83 FOS (0.38) FOSJUNNFKB1NFKB2RELA
SCHEMBL24925661 0.74 P4HA1 (0.38) ALDH1A1MAPTKDM4EL3MBTL1
SCHEMBL10414574 0.74 CA12 (0.54) MAPTRAB9ANPC1HTT
SCHEMBL10414576 0.74 CA12 (0.54) MAPTRAB9ANPC1HTT
SCHEMBL9785541 0.73 SMN1; SMN2 (0.45) FOSJUNNFKB1NFKB2RELA
SCHEMBL2123308 0.72 MAPT (0.50) ALDH1A1MAPTCYP2C9CYP2C19RAB9A
SCHEMBL2666993 0.72 MAPT (0.41) ALDH1A1MAPTDGAT1RAB9ANPSR1
SCHEMBL30272587 0.71 NNMT (0.57) ALDH1A1MAPTKDM4EDGAT1RAB9A
SCHEMBL23200631 0.71 NNMT (0.57) ALDH1A1MAPTKDM4EDGAT1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1019574-B Preparation method with pyrimidine derivatives of desinsection and acaricidal activity ICI PLC (GB) 1992-12-23 CN disclosed
US-5010200-A Insecticide intermediates IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-04-23 US disclosed
US-4962109-A MITICIDES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-10-09 US disclosed
CN-1030412-A PYRIMIDINE DERIVATIVES ICI PLC (GB) 1989-01-18 CN disclosed
EP-0295839-A2 Pyrimidine derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-12-21 EP disclosed