SCHEMBL10654101

SCHEMBL10654101

COCc1ccccc1COC(=O)C(=C(C)C)c1cnc(C(C)(C)C)nc1

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.33
FNTA P49354 1/20 0.32
FNTB P49356 1/20 0.32
PGGT1B P53609 1/20 0.32
HDAC3 O15379 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
MAOB P27338 2/20 0.30
MAOA P21397 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPK1 P28482 1/20 0.30
PKM P14618 1/20 0.30
KMT2A Q03164 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9785451 0.78 FOS (0.38) ALDH1A1PKMKMT2A
SCHEMBL10654105 0.76 GCK (0.33) ALDH1A1MAPK1
SCHEMBL9785488 0.68 KDM4E (0.32) ALDH1A1
SCHEMBL4595467 0.62 MAPK1 (0.52) TDP1ALDH1A1MAPK1KMT2APOLB
SCHEMBL4202389 0.62 TSHR (0.44) TDP1MAOBALDH1A1PKMKMT2A
SCHEMBL29577269 0.62 TSHR (0.44) TDP1MAOBALDH1A1PKMKMT2A
SCHEMBL648491 0.62 IDO1 (0.44) TDP1ALDH1A1KMT2A
SCHEMBL22778456 0.61 RXRA (0.33)
SCHEMBL5255523 0.61 ALDH1A1 (0.65) ALDH1A1PKMKMT2APOLB
SCHEMBL1493636 0.60 TDP1 (0.43) TDP1MAOBMAOAALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0295839-A2 Pyrimidine derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-12-21 EP disclosed