SCHEMBL9789155

SCHEMBL9789155

CC(=O)c1cccc2c1N(N=O)CCC2

nearest known ligand 0.64

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALOX12 P18054 1/20 0.64
ALDH1A1 P00352 3/20 0.42
NOTUM Q6P988 2/20 0.41
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
CES1 P23141 2/20 0.37
DRD2 P14416 1/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
TSHR P16473 1/20 0.37
ATM Q13315 1/20 0.36
LMNA P02545 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
RIPK1 Q13546 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3720316 0.79 NOTUM (0.58) ALOX12ALDH1A1NOTUMKDM4EHPGD
SCHEMBL9789127 0.77 ALOX12 (0.50) ALOX12ALDH1A1KDM4EHPGDMEN1
SCHEMBL8554742 0.75 ALOX12 (0.66) ALOX12ALDH1A1CES1DRD2MEN1
SCHEMBL29785325 0.69 ALOX12 (0.53) ALOX12ALDH1A1KDM4EHPGDCES1
SCHEMBL28890266 0.69 ALOX12 (0.53) ALOX12ALDH1A1KDM4EHPGDCES1
SCHEMBL6643060 0.68 NOTUM (0.44) ALOX12ALDH1A1NOTUMCES1MEN1
SCHEMBL3396949 0.67 ALDH1A1 (0.47) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL1437753 0.67 ALDH1A1 (0.60) ALOX12ALDH1A1NOTUMMEN1KMT2A
SCHEMBL31359858 0.67 BCL2L1 (0.52) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL29933410 0.67 ALDH1A1 (0.60) ALOX12ALDH1A1NOTUMMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4985424-A Certain substituted 1,7-annelated 1h-indazoles being selective antagonists of 5-ht-receptors DUPHAR INTERNATIONAL RESEARCH B.V. (NL) 1991-01-15 US disclosed
US-4950759-A ANTAGONISTS OF NEURONAL 5-HYDROXYTRYPTAMINE(5-HT) RECEPTORS DUPHAR INTERNATIONAL RESEARCH B.V. (NL) 1990-08-21 US disclosed
EP-0350130-A2 New substituted 1,7-annelated 1H-indazoles DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1990-01-10 EP disclosed