SCHEMBL9792898

SCHEMBL9792898

N#Cc1cccc(-c2ccnc(C#N)n2)c1

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.59
CTSS P25774 1/20 0.56
CTSK P43235 1/20 0.56
CLK4 Q9HAZ1 3/20 0.56
GRM5 P41594 5/20 0.55
IDO1 P14902 2/20 0.49
XDH P47989 1/20 0.47
MAOB P27338 1/20 0.45
CYP1A2 P05177 3/20 0.45
CYP3A4 P08684 3/20 0.45
CYP2C19 P33261 3/20 0.45
ALOX15 P16050 2/20 0.45
HSD17B10 Q99714 2/20 0.45
CYP2D6 P10635 2/20 0.45
ALDH1A1 P00352 1/20 0.45
MAPK1 P28482 1/20 0.45
IRAK4 Q9NWZ3 1/20 0.45
LMNA P02545 1/20 0.44
KDM1A O60341 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23662309 0.83 ADORA2A (0.57) KMOCLK4GRM5IDO1XDH
SCHEMBL28844124 0.83 KMO (0.57) KMOCTSSCTSKALDH1A1IRAK4
SCHEMBL7260264 0.83 CLK4 (0.54) KMOCTSSCTSKCLK4GRM5
SCHEMBL1509690 0.81 KMO (0.58) KMOCTSSCTSKCYP1A2CYP2C19
SCHEMBL9792939 0.80 CLK4 (0.62) CLK4GRM5IDO1XDHMAOB
SCHEMBL9792785 0.79 GRM5 (0.50) CTSSCTSKCLK4GRM5IDO1
SCHEMBL25900264 0.79 GRM5 (0.50) CTSSCTSKCLK4GRM5IDO1
SCHEMBL18535 0.79 CTSS (0.63) KMOCTSSCTSKIRAK4
SCHEMBL16395695 0.79 GRM5 (0.66) CLK4GRM5CYP1A2CYP3A4CYP2C19
SCHEMBL4901397 0.78 CLK4 (0.56) CLK4GRM5IDO1XDHCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5064832-A Bipyrimidine Compounds, Antitumor Agents CIBA-GEIGY CORPORATION (US) 1991-11-12 US disclosed
US-4968804-A Bipyridine compounds CIBA-GEIGY CORPORATION (US) 1990-11-06 US disclosed
EP-0350448-A1 Biaryl compounds CIBA-GEIGY AG (CH) 1990-01-10 EP disclosed