SCHEMBL979688

SCHEMBL979688

O=C(Nc1cccc(-c2ccccc2OC(F)(F)F)c1)c1cc2cccc(O)c2oc1=O

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 7/20 0.52
CASP3 P42574 1/20 0.49
ALDH1A1 P00352 1/20 0.49
GLA P06280 1/20 0.49
MAOB P27338 6/20 0.49
AR P10275 2/20 0.47
CBR1 P16152 2/20 0.47
KCNK3 O14649 2/20 0.47
KCNK9 Q9NPC2 2/20 0.47
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
MAOA P21397 2/20 0.46
ADORA3 P0DMS8 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
AKR1C1 Q04828 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL981428 0.94 ALDH1A1 (0.53) CASP3ALDH1A1GLAMAOBKCNK3
SCHEMBL982817 0.91 CASP3 (0.61) CASP3ALDH1A1GLAMAOBKCNK3
SCHEMBL977971 0.85 ALDH1A1 (0.59) CASP3ALDH1A1GLAMAOBKCNK3
SCHEMBL979711 0.85 CASP3 (0.48) CASP3ALDH1A1GLAMAOBKCNK3
SCHEMBL980389 0.82 CASP3 (0.53) CASP3MAOBKCNK3KCNK9NPC1
SCHEMBL979435 0.81 CASP3 (0.49) CASP3ALDH1A1GLAMAOBKCNK3
SCHEMBL979709 0.81 CASP3 (0.53) CASP3MAOBKCNK3KCNK9NPC1
SCHEMBL978586 0.80 ALDH1A1 (0.56) AKR1C3CASP3ALDH1A1GLAMAOB
SCHEMBL980797 0.80 AKR1C3 (0.50) AKR1C3CASP3ALDH1A1GLAMAOB
SCHEMBL980458 0.80 ALDH1A1 (0.55) CASP3ALDH1A1GLAKCNK3KCNK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110021522-A1 ACTIVATORS OF EXECUTIONER PROCASPASES 3, 6 AND 7 THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2011-01-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110021522-A1 ACTIVATORS OF EXECUTIONER PROCASPASES 3, 6 AND 7 CASP7, CASP3, CASP6 AKR1C3 3154/4885CASP3 2/4885ALDH1A1 2806/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.