SCHEMBL9797446

SCHEMBL9797446

CCN(CC)C(=O)COC(=O)c1ccc(N)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.67
CYP1A2 P05177 3/20 0.67
CYP3A4 P08684 3/20 0.67
MAOA P21397 2/20 0.67
TSHR P16473 2/20 0.59
CYP2D6 P10635 2/20 0.59
HTR3A P46098 1/20 0.59
HRH3 Q9Y5N1 1/20 0.59
BLM P54132 1/20 0.57
NPSR1 Q6W5P4 1/20 0.57
CYP2C9 P11712 1/20 0.55
CYP2C19 P33261 1/20 0.55
PDE4D Q08499 1/20 0.55
PHLPP2 Q6ZVD8 1/20 0.54
NPC1 O15118 3/20 0.53
RAB9A P51151 3/20 0.53
MAPT P10636 1/20 0.53
ALDH1A1 P00352 1/20 0.53
SCN1A P35498 2/20 0.51
SCN2A Q99250 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9796885 0.85 ESR1 (0.66) LMNACYP1A2TSHRCYP2D6CYP2C19
Benzoic Acid Diethylcarbamoylmethyl Ester SCHEMBL9653185 0.83 LMNA (0.56) LMNANPC1RAB9AMAPTALDH1A1
SCHEMBL14034893 0.83 LMNA (0.66) LMNACYP1A2CYP3A4MAOATSHR
Benzocaine SCHEMBL1235972 0.81 LMNA (1.00) LMNACYP1A2CYP3A4MAOATSHR
Benzocaine SCHEMBL25100 0.81 LMNA (1.00) LMNACYP1A2CYP3A4MAOATSHR
SCHEMBL11375136 0.80 LMNA (0.77) LMNACYP1A2CYP3A4MAOATSHR
Benzocaine SCHEMBL11021778 0.79 LMNA (0.96) LMNACYP1A2CYP3A4MAOATSHR
Benzocaine SCHEMBL27914401 0.79 LMNA (0.96) LMNACYP1A2CYP3A4MAOATSHR
Benzocaine SCHEMBL15200678 0.79 LMNA (0.96) LMNACYP1A2CYP3A4MAOATSHR
Benzocaine SCHEMBL19031788 0.79 LMNA (0.96) LMNACYP1A2CYP3A4MAOATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5073641-A PRODRUG DERIVATIVES OF CARBOXYLIC ACID DRUGS BUNDGAARD HANS (DK) 1991-12-17 US disclosed
EP-0278977-A1 PRODRUG DERIVATIVES OF CARBOXYLIC ACID DRUGS. BUNDGAARD HANS (DK) 1988-08-24 EP disclosed
WO-1988001615-A1 PRODRUG DERIVATIVES OF CARBOXYLIC ACID DRUGS BUNDGAARD HANS (DK) 1988-03-10 WO disclosed