SCHEMBL9799507

SCHEMBL9799507

CCCCN1CCc2c1c1cccnc1n(-c1ccccc1)c2=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 9/20 0.50
PDE4B Q07343 8/20 0.50
PDE4C Q08493 8/20 0.50
PDE4D Q08499 8/20 0.50
ALDH1A1 P00352 4/20 0.44
TSHR P16473 2/20 0.44
KDM4E B2RXH2 2/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
HPGD P15428 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HSD17B10 Q99714 1/20 0.44
FEN1 P39748 1/20 0.43
L3MBTL1 Q9Y468 2/20 0.40
PDE1A P54750 1/20 0.40
PDE1B Q01064 1/20 0.40
LMNA P02545 1/20 0.40
NPY1R P25929 1/20 0.40
NPY2R P49146 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9799506 0.84 PDE4A (0.54) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL9799632 0.79 FEN1 (0.50) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL9799533 0.77 FEN1 (0.50) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL9799483 0.76 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL9799715 0.74 ALDH1A1 (0.47) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL7278701 0.72 PDE4A (0.87) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL9532938 0.71 FEN1 (0.55) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL9535305 0.71 FEN1 (0.55) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL10378467 0.71 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL9767592 0.70 ALDH1A1 (0.57) PDE4APDE4BPDE4CPDE4DALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4996212-A Antiinflammatory and anti-hyperproliferative compounds SCHERING CORPORATION (US) 1991-02-26 US claimed
US-4996212-A Antiinflammatory and anti-hyperproliferative compounds SCHERING CORPORATION (US) 1991-02-26 US disclosed
US-4859669-A Antiinflammatory and anti-hyperproliferative naphthyridin-4-ones SCHERING CORPORATION (US) 1989-08-22 US disclosed