SCHEMBL9800808

SCHEMBL9800808

CCCCc1ccc(-c2cc(C#N)ccc2OC(=O)C2CCC(C(=O)Oc3ccc(C#N)cc3-c3ccc(CCCC)cc3)CC2)cc1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.45
HSD17B10 Q99714 1/20 0.45
PTGDR2 Q9Y5Y4 1/20 0.42
KDM1A O60341 9/20 0.41
PPARD Q03181 1/20 0.39
PPARA Q07869 1/20 0.39
RARB P10826 1/20 0.38
HRH2 P25021 1/20 0.37
HRH1 P35367 1/20 0.37
ACACB O00763 1/20 0.36
THRA P10827 1/20 0.36
THRB P10828 1/20 0.36
AKR1C2 P52895 1/20 0.36
AKR1C1 Q04828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9800831 0.93 KDM1A (0.47) TSHRHSD17B10PTGDR2KDM1APPARD
SCHEMBL10415568 0.86 RARB (0.41) HSD17B10RARBTHRATHRBAKR1C2
SCHEMBL9800787 0.85 RARB (0.40) HSD17B10PTGDR2RARBTHRATHRB
SCHEMBL9800804 0.84 CTRC (0.44) PTGDR2RARBAKR1C2AKR1C1
SCHEMBL9800791 0.84 FFAR4 (0.49) RARB
SCHEMBL9800817 0.82 RARB (0.45) PPARARARBTHRATHRB
SCHEMBL9800839 0.78 RARB (0.36) TSHRHSD17B10RARBTHRATHRB
SCHEMBL9800824 0.77 FFAR4 (0.51) KDM1A
SCHEMBL11415316 0.77 SPHK1 (0.41)
SCHEMBL9800825 0.76 FFAR4 (0.43) THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0249081-B1 TRANSHEXAHYDROTEREPHTALIC ACID ESTER DERIVATIVES Sato, Hisato (JP) 1991-03-13 EP disclosed
US-4946991-A Liquid ccrystals or their additives SATO HISATO (JP) 1990-08-07 US disclosed