SCHEMBL9806749

SCHEMBL9806749

CCC(C(=O)Nc1ccc2ccn(CCCCCCc3nnn[nH]3)c2c1)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 6/20 0.41
ALDH1A1 P00352 3/20 0.41
ELOVL1 Q9BW60 1/20 0.41
CRHBP P24387 2/20 0.40
CRHR2 Q13324 2/20 0.40
LMNA P02545 2/20 0.40
MAPT P10636 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
HTT P42858 1/20 0.40
KCNQ2 O43526 1/20 0.39
CYP1A2 P05177 1/20 0.39
POLB P06746 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
HDAC3 O15379 3/20 0.39
HDAC4 P56524 3/20 0.39
HDAC7 Q8WUI4 3/20 0.39
HDAC2 Q92769 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9479271 0.81 ALDH1A1 (0.47) HDAC1ALDH1A1ELOVL1CRHBPCRHR2
SCHEMBL9806740 0.80 ADA (0.49) HDAC1LMNAMAPTSMN1; SMN2KCNQ2
SCHEMBL9479139 0.80 ADA (0.49) HDAC1LMNAMAPTSMN1; SMN2KCNQ2
SCHEMBL9490526 0.75 FAAH (0.36) MAPTMEN1KMT2ACYP1A2CYP3A4
SCHEMBL9479257 0.74 KMT2A (0.41) ALDH1A1LMNAMAPTSMN1; SMN2MEN1
SCHEMBL9479222 0.71 MAPT (0.39) HDAC1MAPTMEN1KMT2AHDAC8
SCHEMBL9479523 0.71 MAPT (0.39) HDAC1MAPTMEN1KMT2AHDAC8
SCHEMBL9479635 0.70 MAPT (0.37) HDAC1MAPTMEN1KMT2AHDAC8
SCHEMBL9478509 0.68 MTNR1A (0.32)
SCHEMBL9479109 0.68 ALDH1A1 (0.51) HDAC1ALDH1A1CRHBPCRHR2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997844-A Compounds for the treatment of allergic or inflammatory diseases or shock conditions ICI AMERICAS INC. (US) 1991-03-05 US disclosed
EP-0179619-B1 HETEROCYCLIC AMIDES ICI AMERICAS INC. (US) 1990-09-05 EP disclosed
EP-0179619-A1 Heterocyclic amides ICI AMERICAS INC. (US) 1986-04-30 EP disclosed