SCHEMBL9807589

SCHEMBL9807589

O=C1c2ccccc2CC1C1CCN(CCc2ccc([N+](=O)[O-])cc2)CC1

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 8/20 0.61
HTR2A P28223 8/20 0.61
DRD2 P14416 6/20 0.61
HTR2C P28335 6/20 0.61
HTR2B P41595 6/20 0.61
ACHE P22303 1/20 0.57
KCNJ1 P48048 6/20 0.55
KCNH2 Q12809 5/20 0.55
HRH3 Q9Y5N1 1/20 0.53
ABCB1 P08183 1/20 0.48
ABCG2 Q9UNQ0 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9593183 0.99 SIGMAR1 (0.60) SIGMAR1HTR2ADRD2HTR2CHTR2B
Hydrochloric Acid SCHEMBL9592660 0.99 SIGMAR1 (0.60) SIGMAR1HTR2ADRD2HTR2CHTR2B
SCHEMBL9807598 0.80 SIGMAR1 (0.58) SIGMAR1HTR2ADRD2HTR2CHTR2B
Hydrochloric Acid SCHEMBL9591965 0.79 DRD2 (0.57) SIGMAR1HTR2ADRD2HTR2CHTR2B
SCHEMBL9590736 0.79 KCNJ1 (0.56) SIGMAR1HTR2ADRD2HTR2CHTR2B
SCHEMBL9592696 0.77 DRD2 (0.43) SIGMAR1HTR2ADRD2HTR2CHTR2B
SCHEMBL9807610 0.76 ACHE (0.60) SIGMAR1HTR2ADRD2HTR2CHTR2B
Hydrochloric Acid SCHEMBL9590262 0.75 ACHE (0.58) SIGMAR1HTR2ADRD2HTR2CHTR2B
SCHEMBL5871187 0.75 KCNJ1 (0.56) SIGMAR1HTR2AKCNJ1KCNH2HRH3
SCHEMBL9592259 0.74 ACHE (1.00) SIGMAR1HTR2ADRD2HTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5032598-A Nitrogens containing heterocyclic compounds as class III antiarrhythmic agents MERCK & CO., INC. (US) 1991-07-16 US claimed
EP-0431945-A2 Antiarrhythmic agents MERCK & CO. INC. (US) 1991-06-12 EP claimed