SCHEMBL9807598

SCHEMBL9807598

CS(=O)(=O)Nc1ccc(CCN2CCC(C3Cc4ccccc4C3=O)CC2)cc1

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 12/20 0.58
DRD2 P14416 11/20 0.58
HTR2A P28223 11/20 0.58
HTR2C P28335 11/20 0.58
HTR2B P41595 11/20 0.58
ACHE P22303 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9591965 0.99 DRD2 (0.57) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL9807574 0.91 DRD2 (0.47) SIGMAR1DRD2HTR2AHTR2CHTR2B
Hydrochloric Acid SCHEMBL9592944 0.90 DRD2 (0.46) SIGMAR1DRD2HTR2AHTR2CHTR2B
Methyl Alcohol SCHEMBL9591993 0.88 DRD2 (0.45) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL9807589 0.80 SIGMAR1 (0.61) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL9590055 0.80 DRD2 (0.51) SIGMAR1DRD2HTR2AHTR2CHTR2B
Hydrochloric Acid SCHEMBL9592660 0.79 SIGMAR1 (0.60) SIGMAR1DRD2HTR2AHTR2CHTR2B
Hydrochloric Acid SCHEMBL9593183 0.79 SIGMAR1 (0.60) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL9593272 0.79 ADRA1D (0.57) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL9733215 0.79 KCNH2 (0.59) SIGMAR1DRD2HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5032598-A Nitrogens containing heterocyclic compounds as class III antiarrhythmic agents MERCK & CO., INC. (US) 1991-07-16 US claimed
EP-0431945-A2 Antiarrhythmic agents MERCK & CO. INC. (US) 1991-06-12 EP claimed