SCHEMBL9808975

SCHEMBL9808975

Nc1ccc(Cl)c(-c2ccc([S+]([O-])c3ccc(-c4cc(N)ccc4Cl)cc3)cc2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.42
TSHR P16473 3/20 0.42
PLA2G7 Q13093 1/20 0.39
USP28 Q96RU2 1/20 0.35
AHR P35869 2/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
ALDH1A1 P00352 5/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MAOB P27338 2/20 0.32
HPGD P15428 3/20 0.31
HSD17B10 Q99714 3/20 0.31
MAPT P10636 3/20 0.31
KDM4E B2RXH2 2/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
ALOX15 P16050 2/20 0.31
MAPK1 P28482 1/20 0.31
NPC1 O15118 1/20 0.31
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21021636 0.76 ESR2 (0.50) CYP3A4TSHRPLA2G7CA1CA2
SCHEMBL21021252 0.76 PLA2G7 (0.50) CYP3A4TSHRPLA2G7USP28AHR
SCHEMBL13365533 0.75 CYP2A6 (0.54) CYP3A4TSHRPLA2G7ALDH1A1SMN1; SMN2
SCHEMBL31374861 0.75 CYP2A6 (0.54) CYP3A4TSHRPLA2G7ALDH1A1SMN1; SMN2
SCHEMBL9808973 0.73 HSD17B10 (0.51) CYP3A4ALDH1A1HSD17B10MAPTKDM4E
SCHEMBL2807338 0.73 CYP3A4 (0.65) CYP3A4TSHRPLA2G7CA1CA2
SCHEMBL14744471 0.72 IMPDH2 (0.49) CYP3A4TSHRPLA2G7ALDH1A1SMN1; SMN2
SCHEMBL12458455 0.71 ALDH1A1 (0.47) CYP3A4TSHRPLA2G7USP28AHR
SCHEMBL9629264 0.71 HTR2B (0.50) CYP3A4TSHRUSP28AHRALDH1A1
SCHEMBL310582 0.71 MEN1 (0.50) CYP3A4TSHRCA1CA2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4985463-A Aminodiaryl sulfoxide derivatives, process for their preparation and pharmaceutical and pesticidal compositions containing them RICHTER GEDEON VEGYESZETI GYAR RT (HU) 1991-01-15 US disclosed
US-4831194-A Process for the preparation of nitrodiaryl sulfoxides RICHTER GEDEON VEGYESZETI GYAR RT. (HU) 1989-05-16 US disclosed
US-4710323-A Nitrodiaryl sulfoxide derivatives, process for their preparation and pharmaceutical and pesticidal compositions containing them as active ingredient RICHTER GEDEON VEGYESZETI GYAR RT (HU) 1987-12-01 US disclosed