SCHEMBL9814112

SCHEMBL9814112

COc1ccc2c(c1OCc1ccccc1)CCCC2C#N

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.45
MAOB P27338 2/20 0.45
KDM1A O60341 1/20 0.45
BCHE P06276 5/20 0.41
KDM4E B2RXH2 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
AGTR2 P50052 4/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
ACHE P22303 1/20 0.39
MEN1 O00255 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
AGTR1 P30556 2/20 0.39
HTR1A P08908 1/20 0.39
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
SIGMAR1 Q99720 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9814140 0.83 PARP1 (0.49) MAOBKDM4ECA1CA2ACHE
SCHEMBL6520422 0.82 MAOA (0.53) MAOAMAOBL3MBTL1MEN1KMT2A
SCHEMBL9814134 0.76 CA1 (0.51) CA1CA2SIGMAR1
SCHEMBL8857004 0.74 ADRA1A (0.43) KDM4ECA1CA2ACHEADRA1A
SCHEMBL10751929 0.74 ADRA1A (0.40) CA1CA2ADRA1ASIGMAR1
SCHEMBL21091907 0.73 KMT2A (0.51) MAOAMAOBKDM1AL3MBTL1MEN1
SCHEMBL21091908 0.73 KMT2A (0.51) MAOAMAOBKDM1AL3MBTL1MEN1
SCHEMBL9814133 0.71 MAOB (0.37) MAOAMAOBACHEHTR1AADRA1D
SCHEMBL5713193 0.70 ALDH1A1 (0.54) MAOAMAOBBCHEKDM4EAGTR2
SCHEMBL8857197 0.70 NPSR1 (0.42) KDM4EL3MBTL1CA1CA2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0166937-B1 ADRENERGIC COMPOUNDS ABBOTT LABORATORIES (US) 1991-08-28 EP disclosed
US-4634705-A Adrenergic amidines ABBOTT LABORATORIES (US) 1987-01-06 US disclosed
EP-0166937-A2 Adrenergic compounds ABBOTT LABORATORIES (US) 1986-01-08 EP disclosed