SCHEMBL9817819

SCHEMBL9817819

O=C1CC(c2ccccc2)Sc2ccccc2N1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 1.00
HSD17B10 Q99714 3/20 1.00
TSHR P16473 1/20 1.00
SMN1; SMN2 Q16637 1/20 1.00
MAPK1 P28482 2/20 0.78
GAA P10253 2/20 0.78
TP53 P04637 1/20 0.78
BRD4 O60885 5/20 0.64
CREBBP Q92793 5/20 0.64
MEN1 O00255 3/20 0.63
KMT2A Q03164 3/20 0.63
HPGD P15428 2/20 0.51
KDM4E B2RXH2 1/20 0.51
USP2 O75604 1/20 0.51
ESR1 P03372 1/20 0.51
POLB P06746 1/20 0.51
THRB P10828 1/20 0.51
ALOX15 P16050 1/20 0.51
PTPN7 P35236 1/20 0.51
RECQL P46063 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9602657 0.84 SMN1; SMN2 (0.72) ALDH1A1HSD17B10TSHRSMN1; SMN2MAPK1
SCHEMBL9628805 0.84 HSD17B10 (0.72) ALDH1A1HSD17B10TSHRSMN1; SMN2MAPK1
SCHEMBL4116168 0.82 ALDH1A1 (0.69) ALDH1A1HSD17B10TSHRSMN1; SMN2MAPK1
SCHEMBL11156685 0.80 ALDH1A1 (0.65) ALDH1A1HSD17B10TSHRSMN1; SMN2MAPK1
SCHEMBL10353022 0.78 ALDH1A1 (0.64) ALDH1A1HSD17B10TSHRSMN1; SMN2MAPK1
SCHEMBL14273765 0.78 ALDH1A1 (0.64) ALDH1A1HSD17B10TSHRSMN1; SMN2MAPK1
SCHEMBL11069336 0.78 BRD4 (0.66) ALDH1A1HSD17B10TSHRSMN1; SMN2MAPK1
SCHEMBL8853797 0.78 CREBBP (1.00) ALDH1A1HSD17B10TSHRSMN1; SMN2MAPK1
SCHEMBL10353037 0.78 BRD4 (0.66) ALDH1A1HSD17B10TSHRSMN1; SMN2MAPK1
Bromide SCHEMBL6210437 0.77 ALDH1A1 (0.62) ALDH1A1HSD17B10TSHRSMN1; SMN2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0324181-B1 PROCESS FOR THE PREPARATION OF BENZOTHIAZEPINONE DERIVATIVES BAYER AG (DE) 1991-11-27 EP disclosed
US-4948886-A Process for the preparation of benzothiazepinone derivatives BAYER AKTIENGESELLSCHAFT (DE) 1990-08-14 US disclosed
EP-0292824-B1 PROCESS FOR THE NUCLEAR CHLORINATION OF AROMATIC HYDROCARBONS BAYER AG (DE) 1990-08-01 EP disclosed
US-4851596-A Process for nucleus-chlorination of aromatic hydrocarbons BAYER AKTIENGESELLSCHAFT (DE) 1989-07-25 US disclosed
EP-0324181-A1 Process for the preparation of benzothiazepinone derivatives BAYER AG (DE) 1989-07-19 EP disclosed
EP-0292824-A1 Process for the nuclear chlorination of aromatic hydrocarbons BAYER AG (DE) 1988-11-30 EP disclosed
US-4232027-A ANTIINFLAMMATORY AGENTS E. R. SQUIBB & SONS, INC. (US) 1980-11-04 US disclosed
US-3983106-A ANTIINFLAMMATORY AGENTS E. R. SQUIBB & SONS, INC. (US) 1976-09-28 US disclosed
US-3953469-A TRANQUILLIZERS E. R. SQUIBB & SONS, INC. (US) 1976-04-27 US disclosed
US-3948889-A CHEMICAL INTERMEDIATES E. R. SQUIBB & SONS, INC. (US) 1976-04-06 US disclosed