SCHEMBL9819124

SCHEMBL9819124

N#CC(C(=O)Nc1ccc(C(F)(F)F)cc1)C(=O)c1ccc(Cl)cc1Cl

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 1/20 0.52
P2RX1 P51575 2/20 0.49
P2RX4 Q99571 2/20 0.49
P2RX7 Q99572 2/20 0.49
TMPRSS4 Q9NRS4 2/20 0.49
IDO1 P14902 1/20 0.47
LMNA P02545 4/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ALDH1A1 P00352 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
MAPT P10636 2/20 0.42
HTT P42858 1/20 0.42
JAK2 O60674 2/20 0.41
JAK1 P23458 2/20 0.41
TYK2 P29597 2/20 0.41
CNR2 P34972 1/20 0.41
EPHX2 P34913 1/20 0.40
CLPP Q16740 1/20 0.40
CHRNA7 P36544 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9819107 0.89 GRIK1 (0.50) GRIK1P2RX1P2RX4P2RX7TMPRSS4
SCHEMBL9819165 0.83 RHOC (0.49) GRIK1P2RX1P2RX4P2RX7TMPRSS4
SCHEMBL9818823 0.83 RHOC (0.49) GRIK1P2RX1P2RX4P2RX7TMPRSS4
SCHEMBL9819122 0.82 IDO1 (0.47) GRIK1P2RX1P2RX4P2RX7TMPRSS4
SCHEMBL9818991 0.82 IDO1 (0.49) GRIK1P2RX1P2RX4P2RX7TMPRSS4
SCHEMBL9819209 0.81 IDO1 (0.47) IDO1LMNAMEN1KMT2AMAPT
SCHEMBL9818887 0.80 IDO1 (0.47) GRIK1IDO1ALDH1A1MEN1KMT2A
SCHEMBL9818928 0.79 EPHX2 (0.50) IDO1EPHX2
SCHEMBL9819335 0.78 IDO1 (0.50) IDO1LMNASMN1; SMN2ALDH1A1MEN1
SCHEMBL9819198 0.78 ENPP3 (0.49) IDO1LMNASMN1; SMN2ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5034410-A Nitrile and oxo containing amides or thioamides SYNTEX (U.S.A.) INC. (US) 1991-07-23 US disclosed