SCHEMBL9818928

SCHEMBL9818928

N#CC(C(=O)Nc1ccc(C(F)(F)F)cc1)C(=O)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 2/20 0.50
TRPV1 Q8NER1 3/20 0.49
PTGS1 P23219 2/20 0.49
RORC P51449 1/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
GSK3B P49841 1/20 0.47
DHODH Q02127 1/20 0.47
RAPGEF3 O95398 1/20 0.45
RAPGEF4 Q8WZA2 1/20 0.45
CES2 O00748 1/20 0.45
CES1 P23141 1/20 0.45
KIF11 P52732 1/20 0.44
TGM2 P21980 1/20 0.44
IDO1 P14902 1/20 0.44
KCNQ3 O43525 1/20 0.44
KCNQ2 O43526 1/20 0.44
KCNE1 P15382 1/20 0.44
KCNQ1 P51787 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9818907 0.96 MAOB (0.47) EPHX2TRPV1PTGS1RORCNPC1
SCHEMBL9819042 0.96 MAOB (0.47) EPHX2TRPV1PTGS1RORCNPC1
SCHEMBL9819128 0.94 GSK3B (0.46) EPHX2TRPV1PTGS1RORCNPC1
SCHEMBL9819082 0.94 TRPV1 (0.60) EPHX2TRPV1PTGS1RORCNPC1
SCHEMBL9818823 0.94 RHOC (0.49) EPHX2TRPV1PTGS1NPC1RAB9A
SCHEMBL9819032 0.94 MLYCD (0.52) EPHX2TRPV1PTGS1RORCNPC1
SCHEMBL9818942 0.94 GSK3B (0.46) EPHX2TRPV1PTGS1RORCNPC1
SCHEMBL9819165 0.94 RHOC (0.49) EPHX2TRPV1PTGS1NPC1RAB9A
SCHEMBL9818938 0.94 TRPV1 (0.47) EPHX2TRPV1PTGS1RORCNPC1
SCHEMBL9819035 0.94 MLYCD (0.52) EPHX2TRPV1PTGS1RORCNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5034410-A Nitrile and oxo containing amides or thioamides SYNTEX (U.S.A.) INC. (US) 1991-07-23 US claimed
US-5034410-A Nitrile and oxo containing amides or thioamides SYNTEX (U.S.A.) INC. (US) 1991-07-23 US disclosed