SCHEMBL9819216

SCHEMBL9819216

N#Cc1ccc(C(=O)C(C#N)C(=O)Nc2ccc(C(F)(F)F)c([N+](=O)[O-])c2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 9/20 0.47
CYP3A4 P08684 2/20 0.47
CES2 O00748 1/20 0.47
ABCB11 O95342 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
CYP1A2 P05177 1/20 0.47
GLA P06280 1/20 0.47
ADORA3 P0DMS8 1/20 0.47
CHRM1 P11229 1/20 0.47
CYP2C9 P11712 1/20 0.47
ALOX15 P16050 1/20 0.47
TSHR P16473 1/20 0.47
TBXA2R P21731 1/20 0.47
AADAC P22760 1/20 0.47
MAPK1 P28482 1/20 0.47
CYP2C19 P33261 1/20 0.47
ADRA1A P35348 1/20 0.47
HTT P42858 1/20 0.47
HTR6 P50406 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9819219 0.91 AR (0.48) ARCYP3A4CES2ABCB11ALDH1A1
SCHEMBL9818871 0.83 AR (0.59) ARCYP3A4CES2ABCB11ALDH1A1
SCHEMBL9819190 0.82 AR (0.58) ARCYP3A4CES2ABCB11ALDH1A1
SCHEMBL9819035 0.78 MLYCD (0.52) MLYCDTRPV1KIF11
SCHEMBL9819032 0.78 MLYCD (0.52) MLYCDTRPV1KIF11
SCHEMBL9819414 0.78 LMNA (0.45) ARCYP3A4CES2ABCB11ALDH1A1
SCHEMBL9819214 0.78 GSK3B (0.51) ALDH1A1LMNATSHRMAPK1HTT
SCHEMBL9819097 0.76 P2RX1 (0.50) CYP3A4ALDH1A1LMNACYP1A2CYP2C9
SCHEMBL9818865 0.75 ABCG2 (0.50) ALDH1A1LMNAMAPK1HTTSMN1; SMN2
SCHEMBL9818946 0.75 ABCG2 (0.50) ALDH1A1LMNAMAPK1HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5034410-A Nitrile and oxo containing amides or thioamides SYNTEX (U.S.A.) INC. (US) 1991-07-23 US disclosed