SCHEMBL9819035

SCHEMBL9819035

N#Cc1ccc(NC(=O)C(C#N)C(=O)c2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 1/20 0.52
EPHX2 P34913 3/20 0.45
KIF11 P52732 1/20 0.44
TRPV1 Q8NER1 3/20 0.44
PTGS1 P23219 2/20 0.44
RXFP1 Q9HBX9 1/20 0.43
VNN1 O95497 1/20 0.43
RORC P51449 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
DHODH Q02127 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
GSK3B P49841 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9819032 1.00 MLYCD (0.52) MLYCDEPHX2KIF11TRPV1PTGS1
SCHEMBL9818928 0.94 EPHX2 (0.50) EPHX2KIF11TRPV1PTGS1RORC
SCHEMBL9818907 0.90 MAOB (0.47) EPHX2TRPV1PTGS1RORCNPC1
SCHEMBL9819042 0.90 MAOB (0.47) EPHX2TRPV1PTGS1RORCNPC1
SCHEMBL9819214 0.89 GSK3B (0.51) MLYCDNPC1RAB9AGSK3B
SCHEMBL9818938 0.88 TRPV1 (0.47) EPHX2TRPV1PTGS1RORCNPC1
SCHEMBL9819082 0.88 TRPV1 (0.60) MLYCDEPHX2TRPV1PTGS1RORC
SCHEMBL9819128 0.88 GSK3B (0.46) EPHX2TRPV1PTGS1RORCNPC1
SCHEMBL9819165 0.88 RHOC (0.49) EPHX2TRPV1PTGS1NPC1RAB9A
SCHEMBL9818942 0.88 GSK3B (0.46) EPHX2TRPV1PTGS1RORCNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5034410-A Nitrile and oxo containing amides or thioamides SYNTEX (U.S.A.) INC. (US) 1991-07-23 US disclosed