SCHEMBL9818946

SCHEMBL9818946

N#CC(C(=O)Nc1ccc([N+](=O)[O-])cc1)C(=O)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 1/20 0.50
MEN1 O00255 8/20 0.45
KMT2A Q03164 8/20 0.45
MAPT P10636 6/20 0.45
ALDH1A1 P00352 2/20 0.45
MITF O75030 2/20 0.44
POLB P06746 2/20 0.44
MAPK1 P28482 2/20 0.44
NPC1 O15118 3/20 0.43
RAB9A P51151 2/20 0.43
HTT P42858 1/20 0.43
LMNA P02545 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
PHGDH O43175 1/20 0.42
PKM P14618 1/20 0.42
HPGD P15428 1/20 0.42
PIN1 Q13526 1/20 0.41
EPHX2 P34913 1/20 0.40
TRPV1 Q8NER1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9818865 1.00 ABCG2 (0.50) ABCG2MEN1KMT2AMAPTALDH1A1
SCHEMBL9818928 0.89 EPHX2 (0.50) NPC1RAB9AEPHX2TRPV1
SCHEMBL9819417 0.87 KIF11 (0.50) ABCG2MEN1KMT2AMAPTMITF
SCHEMBL9819349 0.87 MEN1 (0.50) ABCG2MEN1KMT2AMAPTALDH1A1
SCHEMBL9819042 0.86 MAOB (0.47) MEN1KMT2AMITFNPC1RAB9A
SCHEMBL9818907 0.86 MAOB (0.47) MEN1KMT2AMITFNPC1RAB9A
SCHEMBL9819219 0.84 AR (0.48) MEN1KMT2AMAPTALDH1A1POLB
SCHEMBL9818871 0.84 AR (0.59) MAPTALDH1A1MAPK1HTTLMNA
SCHEMBL9819032 0.83 MLYCD (0.52) NPC1RAB9ARXFP1EPHX2TRPV1
SCHEMBL9819165 0.83 RHOC (0.49) MEN1KMT2ANPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5034410-A Nitrile and oxo containing amides or thioamides SYNTEX (U.S.A.) INC. (US) 1991-07-23 US disclosed