SCHEMBL9820846

SCHEMBL9820846

CC1CN(C(=O)C2CC2c2ccc(C(C)(C)C)cc2)CC(C)O1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 6/20 0.47
CRHBP P24387 1/20 0.46
CRHR2 Q13324 1/20 0.46
TRPV1 Q8NER1 1/20 0.45
CNR1 P21554 1/20 0.44
KCNH2 Q12809 1/20 0.44
SIGMAR1 Q99720 4/20 0.42
NPC1 O15118 2/20 0.41
HTT P42858 2/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
NR2F2 P24468 1/20 0.41
RAB9A P51151 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
SLC6A2 P23975 1/20 0.41
HSD17B10 Q99714 1/20 0.40
EBP Q15125 1/20 0.40
MGLL Q99685 1/20 0.40
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9820772 0.82 NPC1 (0.44) HRH3SIGMAR1NPC1HSD17B10
SCHEMBL10683557 0.78 HRH3 (0.39) HRH3CRHBPCRHR2NPC1HSD17B10
SCHEMBL10684339 0.78 HRH3 (0.39) HRH3CRHBPCRHR2NPC1HSD17B10
SCHEMBL10684334 0.77 SMN1; SMN2 (0.38) HRH3CRHBPCRHR2NPC1HTT
SCHEMBL10683685 0.77 SMN1; SMN2 (0.38) HRH3CRHBPCRHR2NPC1HTT
SCHEMBL18216835 0.76 CRHBP (0.71) CRHBPCRHR2NPC1HTTRAB9A
SCHEMBL301271 0.75 FFAR1 (0.55) HRH3TRPV1NPC1HTTLMNA
SCHEMBL1474207 0.75 FFAR1 (0.55) HRH3TRPV1NPC1HTTLMNA
SCHEMBL9820868 0.75 TRPV1 (0.50) HRH3TRPV1NPC1HTTLMNA
SCHEMBL10288267 0.75 FFAR1 (0.55) HRH3TRPV1NPC1HTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0188887-B1 TERTIARY AMINE COMPOUNDS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-05-02 EP disclosed
EP-0251466-A2 Chemical process for the preparation of esters of substituted cyclopropyl caboxylic acids IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-01-07 EP disclosed
EP-0188887-A1 Tertiary amine compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1986-07-30 EP disclosed