SCHEMBL9823140

SCHEMBL9823140

CC(=O)c1ccc(C#CCNCc2ccc3nc[nH]c(=O)c3c2)cc1

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.57
DHFR P00374 6/20 0.55
IP6K1 Q92551 5/20 0.46
IP6K3 Q96PC2 2/20 0.46
IP6K2 Q9UHH9 2/20 0.46
PDPK1 O15530 1/20 0.46
FPGS Q05932 2/20 0.41
PARP1 P09874 6/20 0.41
CHEK1 O14757 1/20 0.38
PIM1 P11309 1/20 0.38
AKT1 P31749 1/20 0.38
FLT3 P36888 1/20 0.38
PIM3 Q86V86 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9823121 0.87 PDPK1 (0.46) SLC2A1DHFRIP6K1IP6K3IP6K2
SCHEMBL9823450 0.82 IP6K1 (0.47) SLC2A1DHFRIP6K1IP6K3IP6K2
SCHEMBL9823281 0.82 DHFR (0.56) DHFRFPGS
SCHEMBL10584902 0.81 MMP13 (0.44) IP6K1PDPK1
SCHEMBL9823195 0.72 DHFR (0.45) DHFRFPGS
SCHEMBL9823134 0.71 DHFR (1.00) SLC2A1DHFR
SCHEMBL9514916 0.70 IP6K1 (0.52) SLC2A1IP6K1IP6K3IP6K2PARP1
SCHEMBL9823278 0.70 DHFR (0.47) DHFRFPGS
SCHEMBL9371240 0.69 IP6K1 (0.61) SLC2A1DHFRIP6K1IP6K3IP6K2
SCHEMBL9823104 0.68 DHFR (0.44) DHFRFPGS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0426666-A1 SUBSTITUTED QUINAZOLINONES AS ANTICANCER AGENTS WARNER-LAMBERT COMPANY (US) 1991-05-15 EP claimed
US-4857530-A THYMIDYLATE SYNTHASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1989-08-15 US claimed
WO-1989004307-A1 SUBSTITUTED QUINAZOLINONES AS ANTICANCER AGENTS WARNER-LAMBERT COMPANY (US) 1989-05-18 WO claimed
EP-0426666-A1 SUBSTITUTED QUINAZOLINONES AS ANTICANCER AGENTS WARNER-LAMBERT COMPANY (US) 1991-05-15 EP disclosed
US-4857530-A THYMIDYLATE SYNTHASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1989-08-15 US disclosed
EP-0316657-A1 Substituted quinazolinones as anticancer agents WARNER-LAMBERT COMPANY (US) 1989-05-24 EP disclosed
WO-1989004307-A1 SUBSTITUTED QUINAZOLINONES AS ANTICANCER AGENTS WARNER-LAMBERT COMPANY (US) 1989-05-18 WO disclosed