SCHEMBL9823322

SCHEMBL9823322

C#CCNc1ccc(C(=O)CCN(CC)CC)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 4/20 0.42
THRA P10827 4/20 0.42
MAPT P10636 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
ALDH1A1 P00352 2/20 0.41
NFKB1 P19838 1/20 0.41
KCNH2 Q12809 1/20 0.41
MMP9 P14780 1/20 0.40
MMP13 P45452 1/20 0.40
ADAM17 P78536 1/20 0.40
TERT O14746 5/20 0.40
POLB P06746 2/20 0.40
CYP3A4 P08684 1/20 0.40
BLM P54132 1/20 0.40
ATM Q13315 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HDAC3 O15379 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9823125 0.92 L3MBTL1 (0.45) THRBTHRAMAPTCA12CA1
SCHEMBL9823319 0.81 ALDH1A1 (0.65) THRBCA12CA9ALDH1A1NFKB1
SCHEMBL17549669 0.75 KMT2A (0.56) THRBTHRAMAPTALDH1A1ATM
SCHEMBL5953952 0.73 GSK3B (0.53) THRBTHRAMAPTALDH1A1SMN1; SMN2
SCHEMBL5954012 0.73 HTR7 (0.61) THRBTHRAMAPTALDH1A1POLB
SCHEMBL9491562 0.73 LMNA (0.59) THRBTHRAMAPTALDH1A1KCNH2
SCHEMBL4817527 0.73 MAPT (0.51) MAPTCA12CA1CA2CA9
SCHEMBL432166 0.73 CA1 (0.51) MAPTCA12CA1CA2CA9
SCHEMBL6322827 0.73 KMT2A (0.67) THRBTHRAMAPTALDH1A1POLB
SCHEMBL9823289 0.72 CA1 (0.54) MAPTCA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0426666-A1 SUBSTITUTED QUINAZOLINONES AS ANTICANCER AGENTS WARNER-LAMBERT COMPANY (US) 1991-05-15 EP disclosed
US-4857530-A THYMIDYLATE SYNTHASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1989-08-15 US disclosed
EP-0316657-A1 Substituted quinazolinones as anticancer agents WARNER-LAMBERT COMPANY (US) 1989-05-24 EP disclosed
WO-1989004307-A1 SUBSTITUTED QUINAZOLINONES AS ANTICANCER AGENTS WARNER-LAMBERT COMPANY (US) 1989-05-18 WO disclosed