SCHEMBL9824624

SCHEMBL9824624

COC(=O)C1=C(C)NC(C)=C(C(=O)OC)C1c1cc(S(C)(=O)=O)ccc1OCCCCN

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 3/20 0.42
OPRM1 P35372 3/20 0.42
KCNH2 Q12809 3/20 0.42
MAPT P10636 2/20 0.42
KDM4E B2RXH2 2/20 0.42
KCNK2 O95069 2/20 0.42
ABCB11 O95342 2/20 0.42
ADORA3 P0DMS8 2/20 0.42
HTR2C P28335 2/20 0.42
HTR2B P41595 2/20 0.42
CACNA1C Q13936 2/20 0.42
SCN5A Q14524 2/20 0.42
ABCC4 O15439 1/20 0.42
PLIN1 O60240 1/20 0.42
CACNA1F O60840 1/20 0.42
GMNN O75496 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GSR P00390 1/20 0.42
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9824685 0.91 MAPT (0.43) DRD1OPRM1KCNH2MAPTKDM4E
SCHEMBL10689136 0.83 HSD17B10 (0.51) DRD1OPRM1KCNH2MAPTKDM4E
SCHEMBL7287257 0.82 ADORA3 (0.53) DRD1OPRM1KCNH2MAPTKDM4E
SCHEMBL10686314 0.79 ATM (0.44) MAPTCYP1A2CYP3A4CYP2D6ADRA2A
SCHEMBL10628072 0.76 ADORA3 (0.48) DRD1OPRM1KCNH2MAPTKDM4E
SCHEMBL9825000 0.76 ADORA3 (0.54) DRD1OPRM1KCNH2MAPTKDM4E
SCHEMBL10488355 0.74 ADORA3 (0.53) DRD1OPRM1KCNH2MAPTKDM4E
SCHEMBL10693040 0.73 CACNA1C (0.64) MAPTADORA3CACNA1CCACNA1FALDH1A1
SCHEMBL9789920 0.73 ADORA3 (0.52) DRD1OPRM1KCNH2MAPTKDM4E
SCHEMBL10688906 0.73 ALDH1A1 (0.42) MAPTKDM4EALDH1A1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0167371-B1 DIHYDROPYRIDINE COMPOUNDS, THEIR PRODUCTION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1991-03-06 EP disclosed
US-4727082-A CARDIOVASCULAR DISORDERS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1988-02-23 US disclosed
EP-0167371-A2 Dihydropyridine compounds, their production, and pharmaceutical compositions containing them YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1986-01-08 EP disclosed