SCHEMBL9826864

SCHEMBL9826864

CC(CCC/C=C/c1ccccc1)(C(=O)O)c1cccnc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 5/20 0.53
CYP2D6 P10635 2/20 0.45
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 2/20 0.45
CYP1A1 P04798 1/20 0.45
CYP1B1 Q16678 1/20 0.45
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
CHRNB2 P17787 1/20 0.42
CHRNB4 P30926 1/20 0.42
CHRNA3 P32297 1/20 0.42
CHRNA7 P36544 1/20 0.42
CHRNA4 P43681 1/20 0.42
ALOX15 P16050 1/20 0.42
CYP11B1 P15538 2/20 0.41
CYP11B2 P19099 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9826871 1.00 TBXAS1 (0.53) TBXAS1CYP2D6CYP1A2CYP3A4CYP1A1
SCHEMBL8168491 0.82 FAAH (0.54) TBXAS1CYP3A4MEN1KMT2AALOX15
SCHEMBL5497372 0.80 KCNA5 (0.48) TBXAS1CYP1A2CYP3A4NPC1RAB9A
SCHEMBL8461392 0.77 CYP1A2 (0.49) TBXAS1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL10512019 0.77 CYP1A2 (0.49) TBXAS1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL10985939 0.75 TBXAS1 (0.50) TBXAS1CYP2D6CYP1A2CYP3A4CYP1A1
SCHEMBL6178344 0.74 CYP1A2 (0.51) TBXAS1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL28365595 0.74 PPARA (0.62) TBXAS1CYP2C19TDP1
SCHEMBL22775934 0.73 CYP1A2 (0.50) TBXAS1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL20613567 0.73 ACLY (0.54) TBXAS1KMT2ACYP2C19ALOX15KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0111997-B1 VINYL CARBOXYLIC ACID DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1991-04-10 EP disclosed
US-4518602-A Vinyl carboxylic acid derivatives, their production and use as inhibitors of thromboxane synthetase TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1985-05-21 US disclosed
EP-0111997-A2 Vinyl carboxylic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1984-06-27 EP disclosed