SCHEMBL9827709

SCHEMBL9827709

CNc1nc(C)cc(-c2cc3ccccc3[nH]2)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.52
AURKB Q96GD4 1/20 0.52
GSK3B P49841 1/20 0.44
RAB9A P51151 5/20 0.44
NPC1 O15118 4/20 0.44
ESR1 P03372 1/20 0.43
TDP1 Q9NUW8 2/20 0.42
MAPT P10636 5/20 0.41
KDM4E B2RXH2 4/20 0.41
MEN1 O00255 3/20 0.41
ALDH1A1 P00352 3/20 0.41
HPGD P15428 3/20 0.41
KMT2A Q03164 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
USP2 O75604 1/20 0.41
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41
GAA P10253 1/20 0.41
ALOX15 P16050 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22940435 0.73 AURKA (0.59) AURKAAURKBGSK3BRAB9ANPC1
SCHEMBL9827717 0.71 TUBB4A (0.55) GSK3BRAB9ANPC1TDP1MAPT
SCHEMBL20008234 0.70 CYP1A2 (0.49) RAB9ANPC1TDP1MAPTKDM4E
SCHEMBL23641151 0.70 GSK3B (0.62) AURKAAURKBGSK3BRAB9ANPC1
SCHEMBL9828516 0.70 AURKA (0.55) AURKAAURKBGSK3BRAB9ANPC1
SCHEMBL21672916 0.69 EHMT2 (0.53) RAB9ANPC1TDP1MAPTKDM4E
SCHEMBL374022 0.69 RAB9A (0.74) AURKAAURKBGSK3BRAB9ANPC1
SCHEMBL29631691 0.69 RAB9A (0.74) AURKAAURKBGSK3BRAB9ANPC1
SCHEMBL13831039 0.69 AURKA (0.50) AURKAAURKBGSK3BRAB9ANPC1
SCHEMBL24326363 0.68 TDP1 (0.46) RAB9ANPC1TDP1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0422178-A1 PYRIMIDINE DERIVATIVES. ICI PLC (GB) 1991-04-17 EP disclosed