SCHEMBL9828516

SCHEMBL9828516

Cc1nc(N)cc(-c2cc3ccccc3[nH]2)n1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.55
AURKB Q96GD4 1/20 0.55
GSK3B P49841 1/20 0.54
AOC3 Q16853 2/20 0.49
RAB9A P51151 4/20 0.46
NPC1 O15118 3/20 0.46
ESR1 P03372 1/20 0.46
ATP4A P20648 2/20 0.45
ATP4B P51164 2/20 0.45
KDM4E B2RXH2 4/20 0.43
MAPT P10636 4/20 0.43
MEN1 O00255 3/20 0.43
ALDH1A1 P00352 3/20 0.43
HPGD P15428 3/20 0.43
KMT2A Q03164 3/20 0.43
USP2 O75604 1/20 0.43
LMNA P02545 1/20 0.43
POLB P06746 1/20 0.43
GAA P10253 1/20 0.43
ALOX15 P16050 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11895098 0.76 GSK3B (0.62) AURKAAURKBGSK3BAOC3RAB9A
SCHEMBL27109712 0.75 AURKA (0.54) AURKAAURKBGSK3BAOC3RAB9A
SCHEMBL4248803 0.73 GSK3B (0.55) AURKAAURKBGSK3BAOC3RAB9A
SCHEMBL22940435 0.72 AURKA (0.59) AURKAAURKBGSK3BRAB9ANPC1
SCHEMBL23641151 0.72 GSK3B (0.62) AURKAAURKBGSK3BAOC3RAB9A
SCHEMBL1807649 0.71 ATP4A (0.65) AURKAAURKBGSK3BAOC3RAB9A
SCHEMBL29631691 0.71 RAB9A (0.74) AURKAAURKBGSK3BAOC3RAB9A
SCHEMBL374022 0.71 RAB9A (0.74) AURKAAURKBGSK3BAOC3RAB9A
SCHEMBL8265150 0.71 ADORA2A (0.66) RAB9ANPC1KDM4EMAPTMEN1
SCHEMBL693581 0.70 GSK3B (0.59) AURKAAURKBGSK3BRAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0422178-A1 PYRIMIDINE DERIVATIVES. ICI PLC (GB) 1991-04-17 EP disclosed
WO-1990012790-A1 PYRIMIDINE DERIVATIVES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-11-01 WO disclosed