SCHEMBL9828934

SCHEMBL9828934

COc1ccc(CCN(C)CCCCOc2ccc(C3(CCCN(C)C)Sc4ccccc4N(C)C3=O)cc2)cc1OC

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMPD1 P17405 8/20 0.49
ABCB1 P08183 2/20 0.42
SCN1A P35498 1/20 0.42
SCN2A Q99250 1/20 0.42
SCN3A Q9NY46 1/20 0.42
CYP3A4 P08684 2/20 0.40
MAPT P10636 2/20 0.40
KDM4E B2RXH2 1/20 0.40
TP53 P04637 1/20 0.40
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
HCN4 Q9Y3Q4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10672717 0.90 SMPD1 (0.50) SMPD1ABCB1CYP3A4MAPTKDM4E
SCHEMBL9830080 0.85 ALDH1A1 (0.42) SCN1ASCN2ASCN3AMAPTKDM4E
SCHEMBL9829599 0.85 SMPD1 (0.51) SMPD1ABCB1SCN1ASCN2ASCN3A
Hydrochloric Acid SCHEMBL9829648 0.85 BCHE (0.39) SMPD1KDM4E
Hydrochloric Acid SCHEMBL9830009 0.85 SMPD1 (0.51) SMPD1ABCB1CYP3A4MAPTKDM4E
Oxalic Acid SCHEMBL10673157 0.84 SMPD1 (0.49) SMPD1ABCB1CYP3A4MAPTKDM4E
SCHEMBL9830032 0.83 CACNA1B (0.43) SCN1ASCN2ASCN3AMAPTKDM4E
Oxalic Acid SCHEMBL9831243 0.80 SMPD1 (0.47) SMPD1ABCB1SCN1ASCN2ASCN3A
Hydrochloric Acid SCHEMBL9829638 0.80 ALDH1A1 (0.41) SCN1ASCN2ASCN3AMAPTKDM4E
Oxalic Acid SCHEMBL9831824 0.80 SMPD1 (0.46) SMPD1ABCB1SCN1ASCN2ASCN3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0233291-B1 2-ARYLBENZOTHIAZINE DERIVATIVES SANTEN PHARMACEUTICAL CO., LTD. (JP) 1991-03-13 EP disclosed
US-4739050-A CALCIUM ANTAGONIST, ANTICOAGULANT SANTEN PHARMACEUTICAL CO., LTD. (JP) 1988-04-19 US disclosed
EP-0233291-A1 2-ARYLBENZOTHIAZINE DERIVATIVES SANTEN PHARMACEUTICAL CO., LTD. (JP) 1987-08-26 EP disclosed