SCHEMBL9829580

SCHEMBL9829580

Cc1nc(-c2cccc(Cl)c2)oc1COC(C)(C)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
VDR P11473 9/20 0.48
PPARD Q03181 8/20 0.48
SLC16A3 O15427 6/20 0.48
MCTS1 Q9ULC4 3/20 0.48
SLC16A1 P53985 5/20 0.48
IKBKB O14920 1/20 0.46
PPARG P37231 3/20 0.45
PPARA Q07869 3/20 0.45
ESR1 P03372 2/20 0.45
THRA P10827 2/20 0.45
THRB P10828 2/20 0.45
RXRA P19793 2/20 0.45
ESR2 Q92731 2/20 0.45
FFAR1 O14842 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Romazarit SCHEMBL43265 0.86 ALDH1A1 (0.50) PPARDSLC16A3MCTS1SLC16A1IKBKB
SCHEMBL9831905 0.85 NOTUM (0.44) VDRPPARDSLC16A3MCTS1SLC16A1
Romazarit SCHEMBL3226211 0.85 ALDH1A1 (0.49) PPARDSLC16A3MCTS1SLC16A1IKBKB
SCHEMBL9830223 0.79 PPARD (0.50) VDRPPARDSLC16A3MCTS1SLC16A1
SCHEMBL9831350 0.77 PPARD (0.46) VDRPPARDPPARGPPARAFFAR1
SCHEMBL9830285 0.77 PPARD (0.65) PPARDIKBKBPPARGPPARAFFAR1
SCHEMBL9833185 0.77 IKBKB (0.50) VDRPPARDIKBKBPPARGPPARA
SCHEMBL9831640 0.76 ALDH1A1 (0.49) VDRPPARDSLC16A3MCTS1SLC16A1
SCHEMBL9830056 0.75 PPARA (0.50) PPARDSLC16A3MCTS1SLC16A1IKBKB
Romazarit SCHEMBL9831287 0.75 ALDH1A1 (0.48) VDRPPARDSLC16A3MCTS1SLC16A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0220573-B1 HETEROCYCLIC COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 1991-12-11 EP claimed
EP-0220573-B1 HETEROCYCLIC COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 1991-12-11 EP disclosed
US-4774253-A ETHER,-ACIDS, ESTERS OR AMIDES HOFFMANN-LA ROCHE INC. (US) 1988-09-27 US disclosed