SCHEMBL9833185

SCHEMBL9833185

Cc1nc(-c2cccc(Cl)c2)oc1CO

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.50
NPC1 O15118 2/20 0.46
TP53 P04637 2/20 0.46
RAB9A P51151 2/20 0.46
TSHR P16473 1/20 0.46
NFKB1 P19838 1/20 0.46
NFKB2 Q00653 1/20 0.46
RELA Q04206 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
MAOB P27338 1/20 0.45
ALOX15 P16050 1/20 0.45
NOTUM Q6P988 3/20 0.44
MAPT P10636 2/20 0.44
SLC9A1 P19634 1/20 0.44
VDR P11473 3/20 0.42
PPARD Q03181 2/20 0.42
TRPM8 Q7Z2W7 1/20 0.41
ESR1 P03372 1/20 0.41
THRA P10827 1/20 0.41
THRB P10828 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1553828 0.85 NPC1 (0.49) NPC1TP53RAB9ATSHRSMN1; SMN2
SCHEMBL9831245 0.81 KDM4E (0.52) IKBKBNPC1RAB9ATSHRNFKB1
SCHEMBL6377222 0.81 KDM4E (0.51) IKBKBNPC1RAB9ANFKB1NFKB2
SCHEMBL9832652 0.81 NOTUM (0.44) IKBKBNPC1TP53RAB9ASMN1; SMN2
SCHEMBL5536101 0.80 NPC1 (0.53) IKBKBNPC1TP53RAB9ATSHR
SCHEMBL14019461 0.78 ALDH1A1 (0.44) IKBKBNPC1TP53RAB9ATSHR
SCHEMBL25180859 0.77 MAPT (0.54) IKBKBNPC1TP53RAB9ATSHR
SCHEMBL5540607 0.77 NPC1 (0.50) IKBKBNPC1TP53RAB9ATSHR
SCHEMBL9829580 0.77 VDR (0.48) IKBKBVDRPPARDESR1THRA
SCHEMBL8989246 0.74 IKBKB (0.49) IKBKBNPC1TP53RAB9ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0220573-B1 HETEROCYCLIC COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 1991-12-11 EP disclosed
US-4774253-A ETHER,-ACIDS, ESTERS OR AMIDES HOFFMANN-LA ROCHE INC. (US) 1988-09-27 US disclosed
EP-0220573-A1 Heterocyclic compounds F. HOFFMANN-LA ROCHE AG (CH) 1987-05-06 EP disclosed