SCHEMBL9830186

SCHEMBL9830186

Nc1n[nH]cc1C(=O)c1ccccc1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
MAPT P10636 1/20 0.46
CDK2 P24941 2/20 0.45
CCNB2 O95067 1/20 0.45
CCNE2 O96020 1/20 0.45
CDK1 P06493 1/20 0.45
CDK4 P11802 1/20 0.45
CCNB1 P14635 1/20 0.45
CCND1 P24385 1/20 0.45
CCNE1 P24864 1/20 0.45
CCND2 P30279 1/20 0.45
CCND3 P30281 1/20 0.45
CCNB3 Q8WWL7 1/20 0.45
CES2 O00748 1/20 0.44
CES1 P23141 1/20 0.44
ALOX15 P16050 1/20 0.42
KMT2A Q03164 2/20 0.41
CDK5 Q00535 3/20 0.40
CDK5R1 Q15078 3/20 0.40
PKM P14618 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3982930 0.78 MAPT (0.52) ALDH1A1MAPTCDK2CCNB2CCNE2
SCHEMBL30293901 0.76 CES2 (0.71) ALDH1A1MAPTCES2CES1ALOX15
SCHEMBL250099 0.76 CES2 (0.71) ALDH1A1MAPTCES2CES1ALOX15
SCHEMBL9832213 0.75 LTA4H (0.44) ALDH1A1MAPTCDK2CES2CES1
SCHEMBL27185988 0.74 CES2 (0.68) ALDH1A1MAPTCES2CES1ALOX15
Hydrochloric Acid SCHEMBL27733532 0.74 CES2 (0.68) ALDH1A1MAPTCES2CES1ALOX15
SCHEMBL31574193 0.74 CES2 (0.68) ALDH1A1MAPTCES2CES1ALOX15
SCHEMBL9831962 0.74 PARP1 (0.47) ALDH1A1CDK2CDK4CCND1CES2
SCHEMBL5282720 0.73 MAPT (0.59) ALDH1A1MAPTCES2CES1ALOX15
SCHEMBL29664874 0.73 MAPT (0.59) ALDH1A1MAPTCES2CES1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0129846-B1 (3-AMINO-1H-PYRAZOL-4-YL)(ARYL)METHANONES AMERICAN CYANAMID COMPANY (US) 1991-05-08 EP claimed
EP-0129846-A2 (3-Amino-1H-pyrazol-4-yl)(aryl)methanones AMERICAN CYANAMID COMPANY (US) 1985-01-02 EP claimed