SCHEMBL9832213

SCHEMBL9832213

Nc1n[nH]cc1C(=O)c1ccc(F)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.44
MAPK14 Q16539 3/20 0.40
ALDH1A1 P00352 1/20 0.40
HTT P42858 1/20 0.40
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
NPC1 O15118 3/20 0.38
RXFP1 Q9HBX9 1/20 0.38
CCNA2 P20248 1/20 0.38
CDK2 P24941 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CDK5 Q00535 1/20 0.37
CDK5R1 Q15078 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MAPT P10636 1/20 0.37
PKM P14618 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7369952 0.83 ALDH1A1 (0.48) ALDH1A1HTTCES2CES1NPC1
SCHEMBL9832465 0.83 KMT2A (0.49) HTTNPC1MEN1KMT2ARAB9A
SCHEMBL3982930 0.83 MAPT (0.52) MAPK14ALDH1A1CCNA2CDK2MEN1
SCHEMBL9831962 0.81 PARP1 (0.47) MAPK14ALDH1A1HTTCES2CES1
SCHEMBL9830883 0.81 KMT2A (0.44) LTA4HALDH1A1CCNA2CDK2MEN1
SCHEMBL7399203 0.81 NPC1 (0.54) MAPK14ALDH1A1HTTCES2CES1
SCHEMBL9830186 0.75 ALDH1A1 (0.46) MAPK14ALDH1A1CES2CES1NPC1
SCHEMBL5821548 0.74 PTPN1 (0.35) ALDH1A1NPC1MEN1KMT2ARAB9A
SCHEMBL9831766 0.74 TSHR (0.58) ALDH1A1HTTMEN1KMT2ACDK5
SCHEMBL9832146 0.72 SRD5A2 (0.50) ALDH1A1CES2CCNA2CDK2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0129846-B1 (3-AMINO-1H-PYRAZOL-4-YL)(ARYL)METHANONES AMERICAN CYANAMID COMPANY (US) 1991-05-08 EP claimed
EP-0129846-A2 (3-Amino-1H-pyrazol-4-yl)(aryl)methanones AMERICAN CYANAMID COMPANY (US) 1985-01-02 EP claimed
US-4521422-A ANTICONVULSANT, ANTIEPILEPTIC AGENTS, SEDATIVES, MUSCLE RELAXANTS AMERICAN CYANAMID COMPANY (US) 1985-06-04 US disclosed