SCHEMBL9830729

SCHEMBL9830729

CCOC(=O)c1ccc(N2CCC(=O)C2)c(Br)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A1 P18405 1/20 0.47
SRD5A2 P31213 1/20 0.47
PRMT1 Q99873 1/20 0.43
ALDH1A1 P00352 5/20 0.43
RARA P10276 2/20 0.43
RARB P10826 2/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
CA14 Q9ULX7 1/20 0.43
KDM4E B2RXH2 3/20 0.42
MAPK1 P28482 2/20 0.42
POLB P06746 1/20 0.42
ALOX15 P16050 1/20 0.42
HSD17B10 Q99714 1/20 0.42
EGFR P00533 1/20 0.41
MAPT P10636 2/20 0.41
ALOX5 P09917 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9830967 0.88 SRD5A1 (0.49) SRD5A1SRD5A2PRMT1ALDH1A1RARA
SCHEMBL9832862 0.86 ALDH1A1 (0.52) SRD5A1SRD5A2PRMT1ALDH1A1RARA
SCHEMBL9832356 0.85 L3MBTL1 (0.54) SRD5A1SRD5A2ALDH1A1KDM4EMAPK1
SCHEMBL9831632 0.84 HSD17B2 (0.53) SRD5A1SRD5A2PRMT1ALDH1A1RARA
SCHEMBL9831758 0.81 KDM4E (0.42) ALDH1A1KDM4EPOLBMAPTHSP90AA1
SCHEMBL31593035 0.81 WDR5 (0.53) SRD5A1SRD5A2PRMT1ALDH1A1RARA
SCHEMBL28961520 0.80 PRMT1 (0.47) SRD5A1SRD5A2PRMT1ALDH1A1RARA
SCHEMBL9829081 0.79 ALDH1A1 (0.55) ALDH1A1CA12CA1CA2CA7
SCHEMBL9832079 0.79 PDE3B (0.40) SRD5A1SRD5A2ALDH1A1CA12CA1
SCHEMBL9832735 0.76 ALDH1A1 (0.45) SRD5A1SRD5A2ALDH1A1RARARARB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0449989-A1 6,7 DIHYDROPYRROLO 3,4-c] PYRIDO 2,3-d] PYRIMIDINE DERIVATIVES Sloan-Kettering Institute For Cancer Research (US) 1991-10-09 EP claimed
WO-1990007496-A1 6,7 DIHYDROPYRROLO[3,4-c] PYRIDO[2,3-d] PYRIMIDINE DERIVATIVES SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-07-12 WO claimed