SCHEMBL9830732

SCHEMBL9830732

COc1ccc(OCCC=O)c(C2(SC)Sc3ccccc3N(C)C2=O)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADAMTS5 Q9UNA0 1/20 0.36
CYP2C19 P33261 2/20 0.33
CYP2C9 P11712 1/20 0.33
MAPT P10636 7/20 0.33
ALDH1A1 P00352 5/20 0.33
RAB9A P51151 5/20 0.33
KDM4E B2RXH2 4/20 0.33
NPC1 O15118 3/20 0.33
L3MBTL1 Q9Y468 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
PKM P14618 1/20 0.33
TSHR P16473 1/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
NFKB1 P19838 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32
ALOX15 P16050 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9829551 0.89 PTPN1 (0.35) ADAMTS5MAPTALDH1A1RAB9ATSHR
SCHEMBL9831349 0.87 ADAMTS5 (0.34) ADAMTS5MAPTALDH1A1RAB9AKDM4E
SCHEMBL9832228 0.84 ADAMTS5 (0.32) ADAMTS5CYP2C19CYP2C9MAPTALDH1A1
SCHEMBL9828736 0.80 MEN1 (0.44) ADAMTS5CYP2C19MAPTALDH1A1RAB9A
SCHEMBL9829147 0.80 SMPD1 (0.51)
Hydrochloric Acid SCHEMBL9832211 0.80 SMPD1 (0.50) ALOX15
SCHEMBL9828526 0.79 SMPD1 (0.42)
Hydrochloric Acid SCHEMBL9831196 0.79 SMPD1 (0.49) ALOX15
Hydrochloric Acid SCHEMBL9829234 0.79 SMPD1 (0.41)
Hydrochloric Acid SCHEMBL9828653 0.79 BCHE (0.36) MAPTALDH1A1LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0233291-B1 2-ARYLBENZOTHIAZINE DERIVATIVES SANTEN PHARMACEUTICAL CO., LTD. (JP) 1991-03-13 EP disclosed
US-4739050-A CALCIUM ANTAGONIST, ANTICOAGULANT SANTEN PHARMACEUTICAL CO., LTD. (JP) 1988-04-19 US disclosed