SCHEMBL9831375

SCHEMBL9831375

CCC(CC)C1C(=O)Nc2cc3c(cc21)NC(c1cccnc1)N3

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.41
MAPT P10636 6/20 0.41
MAPK1 P28482 4/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
RECQL P46063 1/20 0.41
RAB9A P51151 1/20 0.41
MCL1 Q07820 1/20 0.41
GSK3B P49841 1/20 0.38
ALDH1A1 P00352 6/20 0.37
CYP3A4 P08684 3/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2C19 P33261 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
TSHR P16473 3/20 0.36
CASP1 P29466 1/20 0.35
CASP7 P55210 1/20 0.35
GAA P10253 2/20 0.34
HPGD P15428 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9831225 0.87 KDM4E (0.44) KDM4EMAPTMAPK1MEN1KMT2A
SCHEMBL9831075 0.86 KDM4E (0.40) KDM4EKMT2AALDH1A1TSHRGAA
SCHEMBL9831454 0.81 MAPT (0.42) KDM4EMAPTMAPK1MEN1KMT2A
SCHEMBL9831252 0.78 KDM4E (0.46) KDM4EMAPTMAPK1MEN1KMT2A
SCHEMBL9833862 0.77 KDM4E (0.43) KDM4EMAPTMAPK1MEN1KMT2A
SCHEMBL9833956 0.77 KDM4E (0.52) KDM4EMAPTMAPK1MEN1KMT2A
SCHEMBL10473665 0.76 MAPT (0.42) KDM4EMAPTMAPK1MEN1KMT2A
SCHEMBL9831088 0.76 KDM4E (0.41) KDM4EMAPTMAPK1MEN1KMT2A
SCHEMBL9833436 0.75 BRPF1 (0.30)
SCHEMBL10471544 0.74 MAPT (0.45) KDM4EMAPTMAPK1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161632-B1 PYRROLO-BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1991-04-10 EP disclosed
US-4963686-A INTERMEDIATES FOR INOTROPIC AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1990-10-16 US disclosed