SCHEMBL9831075

SCHEMBL9831075

CCC(CC)C1C(=O)Nc2cc3c(cc21)NC(c1ccncc1)N3

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HSD17B10 Q99714 1/20 0.40
GAA P10253 1/20 0.34
TSHR P16473 1/20 0.34
KMT2A Q03164 1/20 0.34
DDB1 Q16531 1/20 0.30
CRBN Q96SW2 1/20 0.30
PGR P06401 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9831375 0.86 KDM4E (0.41) KDM4EALDH1A1HSD17B10GAATSHR
SCHEMBL9833436 0.82 BRPF1 (0.30)
SCHEMBL9833587 0.79 KDM4E (0.41) KDM4EALDH1A1HSD17B10GAATSHR
SCHEMBL9830572 0.75 ALDH1A1 (0.42) KDM4EALDH1A1HSD17B10GAATSHR
SCHEMBL9833486 0.74 TDP2 (0.45) KDM4EALDH1A1HSD17B10GAATSHR
SCHEMBL9832287 0.74 KDM4E (0.41) KDM4EALDH1A1HSD17B10GAATSHR
SCHEMBL9833215 0.74 ALDH1A1 (0.41) KDM4EALDH1A1HSD17B10GAATSHR
SCHEMBL9832940 0.73 KDM4E (0.49) KDM4EALDH1A1HSD17B10GAATSHR
SCHEMBL10471688 0.73 KDM4E (0.38) KDM4EALDH1A1HSD17B10GAATSHR
SCHEMBL10375402 0.73 TNKS2 (0.42) GAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161632-B1 PYRROLO-BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1991-04-10 EP disclosed
US-4963686-A INTERMEDIATES FOR INOTROPIC AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1990-10-16 US disclosed