SCHEMBL9831487

SCHEMBL9831487

CCOC(=O)c1c(C)cc(N2CCC(=O)C2)cc1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
ALDH1A1 P00352 4/20 0.44
NR1H2 P55055 1/20 0.43
NR1H3 Q13133 1/20 0.43
KCNQ2 O43526 1/20 0.42
USP2 O75604 2/20 0.42
KDM4E B2RXH2 3/20 0.40
MAPT P10636 2/20 0.40
HPGD P15428 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
MAPK1 P28482 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
LMNA P02545 2/20 0.38
GAA P10253 1/20 0.38
CYP1A2 P05177 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9830345 0.86 NR1H2 (0.41) CYP3A4SMN1; SMN2TDP1ALDH1A1NR1H2
SCHEMBL9829312 0.86 MAPT (0.43) CYP3A4SMN1; SMN2TDP1ALDH1A1NR1H2
SCHEMBL9831828 0.86 NR1H2 (0.41) CYP3A4SMN1; SMN2TDP1ALDH1A1NR1H2
SCHEMBL9829593 0.85 KCNK3 (0.40) CYP3A4SMN1; SMN2TDP1ALDH1A1NR1H2
SCHEMBL9830224 0.83 MAPT (0.55) SMN1; SMN2TDP1ALDH1A1USP2KDM4E
SCHEMBL9829081 0.79 ALDH1A1 (0.55) CYP3A4SMN1; SMN2TDP1ALDH1A1HPGD
SCHEMBL9832735 0.76 ALDH1A1 (0.45) ALDH1A1USP2KDM4EMAPTL3MBTL1
SCHEMBL9830612 0.76 MAPT (0.50) ALDH1A1NR1H2NR1H3USP2KDM4E
SCHEMBL9832167 0.76 MAPT (0.50) SMN1; SMN2ALDH1A1USP2KDM4EMAPT
SCHEMBL9830967 0.75 SRD5A1 (0.49) SMN1; SMN2ALDH1A1KDM4EMAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0449989-A1 6,7 DIHYDROPYRROLO 3,4-c] PYRIDO 2,3-d] PYRIMIDINE DERIVATIVES Sloan-Kettering Institute For Cancer Research (US) 1991-10-09 EP claimed
WO-1990007496-A1 6,7 DIHYDROPYRROLO[3,4-c] PYRIDO[2,3-d] PYRIMIDINE DERIVATIVES SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-07-12 WO claimed