SCHEMBL9831983

SCHEMBL9831983

N#CC(C#N)=C1CCCN1CC1CCCCC1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 12/20 0.38
CHRM5 P08912 2/20 0.36
ADRA2C P18825 1/20 0.36
PKM P14618 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRL1 P41146 1/20 0.33
ACHE P22303 1/20 0.33
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
CHRM1 P11229 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9832183 0.71 NOS3 (0.36) HRH3
SCHEMBL10407364 0.70 CHRM5 (0.43) HRH3CHRM5ADRA2COPRM1OPRL1
SCHEMBL4513010 0.68 KDM4E (0.47) CHRM5ADRA2CPKMCHRM2CHRM4
SCHEMBL27975973 0.66 PKM (0.40) HRH3CHRM5ADRA2CPKMACHE
SCHEMBL15319538 0.63 CHRM5 (0.47) HRH3CHRM5ADRA2CACHECHRM2
SCHEMBL14401611 0.62 HRH3 (0.43) HRH3
SCHEMBL1307885 0.61 CHRM5 (0.59) CHRM5ADRA2COPRM1OPRL1ACHE
SCHEMBL7384750 0.60 KDM4E (0.52) CHRM5PKMCHRM2CHRM4CHRM1
SCHEMBL29600183 0.59 ALDH1A1 (0.58) HRH3OPRM1OPRL1CHRM2CHRM4
SCHEMBL1307549 0.59 CHRM5 (0.56) CHRM5ADRA2COPRM1OPRL1ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0449989-A1 6,7 DIHYDROPYRROLO 3,4-c] PYRIDO 2,3-d] PYRIMIDINE DERIVATIVES Sloan-Kettering Institute For Cancer Research (US) 1991-10-09 EP claimed
WO-1990007496-A1 6,7 DIHYDROPYRROLO[3,4-c] PYRIDO[2,3-d] PYRIMIDINE DERIVATIVES SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-07-12 WO claimed