SCHEMBL9832245

SCHEMBL9832245

Cc1c(Cl)ccc(C(=O)OC(C)C)c1NS(=O)(=O)c1nc2nccc(C)n2n1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
MAPK1 P28482 2/20 0.40
KDM4E B2RXH2 1/20 0.40
L3MBTL1 Q9Y468 3/20 0.39
POLB P06746 2/20 0.38
MAPT P10636 2/20 0.37
RXFP1 Q9HBX9 2/20 0.37
SMN1; SMN2 Q16637 4/20 0.36
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
RECQL P46063 1/20 0.35
PKM P14618 1/20 0.35
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9832028 0.91 ALDH1A1 (0.40) ALDH1A1MAPK1KDM4EL3MBTL1POLB
SCHEMBL9832400 0.90 L3MBTL1 (0.40) ALDH1A1MAPK1KDM4EL3MBTL1POLB
SCHEMBL9830619 0.90 ALDH1A1 (0.43) ALDH1A1MAPK1KDM4EL3MBTL1POLB
SCHEMBL9832070 0.89 L3MBTL1 (0.41) ALDH1A1MAPK1KDM4EL3MBTL1POLB
SCHEMBL9831282 0.88 TSHR (0.48) ALDH1A1KDM4EL3MBTL1POLBMAPT
SCHEMBL9832897 0.88 ALDH1A1 (0.49) ALDH1A1MAPK1KDM4EL3MBTL1POLB
SCHEMBL9831782 0.86 ALDH1A1 (0.39) ALDH1A1MAPK1KDM4EL3MBTL1POLB
SCHEMBL10665699 0.85 LMNA (0.42) MAPK1KDM4EL3MBTL1POLBMAPT
SCHEMBL9832089 0.85 L3MBTL1 (0.45) ALDH1A1MAPK1KDM4EL3MBTL1POLB
SCHEMBL9832458 0.84 L3MBTL1 (0.40) ALDH1A1MAPK1KDM4EL3MBTL1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0142152-B1 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1991-03-20 EP claimed
EP-0142152-A2 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1985-05-22 EP claimed
EP-0142152-B1 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1991-03-20 EP disclosed
EP-0217353-B1 SILVER HALIDE COLOR PHOTOGRAPHIC MATERIALS FUJI PHOTO FILM CO., LTD. (JP) 1991-01-16 EP disclosed
EP-0330137-A1 Intermediate compounds for the preparation of 1,2,4-triazolo [1,5-a]pyrimidine-2-sulfonamides DowElanco (US) 1989-08-30 EP disclosed
US-4755212-A Novel substituted 1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonamides and compositions and method for inhibiting pollen formation in corn THE DOW CHEMICAL COMPANY (US) 1988-07-05 US disclosed
US-4741764-A SUPPRESSION OF NITRIFICATION OF AMMONIUM NITROGEN IN THE SOIL THE DOW CHEMICAL COMPANY (US) 1988-05-03 US disclosed
US-4740233-A Substituted 1,2,4-triazolo[1,5-a]-pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1988-04-26 US disclosed
EP-0142152-A2 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1985-05-22 EP disclosed