SCHEMBL9832897

SCHEMBL9832897

CCOC(=O)c1ccc(Cl)c(C)c1NS(=O)(=O)c1nc2nccc(C)n2n1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.49
MAPK1 P28482 2/20 0.45
POLB P06746 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.41
MAPT P10636 2/20 0.41
KDM4E B2RXH2 2/20 0.40
LMNA P02545 1/20 0.40
KMT2A Q03164 2/20 0.40
RECQL P46063 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MCL1 Q07820 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
RXFP1 Q9HBX9 2/20 0.39
TSHR P16473 1/20 0.38
HTT P42858 1/20 0.38
THRB P10828 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9830619 0.91 ALDH1A1 (0.43) ALDH1A1MAPK1POLBL3MBTL1MAPT
SCHEMBL9832261 0.90 ALDH1A1 (0.49) ALDH1A1MAPK1POLBL3MBTL1MAPT
SCHEMBL9830969 0.90 ALDH1A1 (0.51) ALDH1A1MAPK1POLBL3MBTL1MAPT
SCHEMBL9832798 0.89 ALDH1A1 (0.54) ALDH1A1MAPK1POLBL3MBTL1MAPT
SCHEMBL9832245 0.88 ALDH1A1 (0.40) ALDH1A1MAPK1POLBL3MBTL1MAPT
SCHEMBL9832454 0.88 ALDH1A1 (0.49) ALDH1A1MAPK1POLBL3MBTL1KDM4E
SCHEMBL9831782 0.87 ALDH1A1 (0.39) ALDH1A1MAPK1POLBL3MBTL1MAPT
SCHEMBL10666159 0.85 MAPK1 (0.44) ALDH1A1MAPK1MAPTKDM4ELMNA
SCHEMBL9831492 0.84 ALDH1A1 (0.56) ALDH1A1MAPK1POLBL3MBTL1MAPT
SCHEMBL9832683 0.83 ALDH1A1 (0.50) ALDH1A1MAPK1POLBL3MBTL1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0142152-B1 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1991-03-20 EP claimed
EP-0142152-A2 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1985-05-22 EP claimed
EP-0142152-B1 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1991-03-20 EP disclosed
EP-0330137-A1 Intermediate compounds for the preparation of 1,2,4-triazolo [1,5-a]pyrimidine-2-sulfonamides DowElanco (US) 1989-08-30 EP disclosed
US-4755212-A Novel substituted 1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonamides and compositions and method for inhibiting pollen formation in corn THE DOW CHEMICAL COMPANY (US) 1988-07-05 US disclosed
US-4741764-A SUPPRESSION OF NITRIFICATION OF AMMONIUM NITROGEN IN THE SOIL THE DOW CHEMICAL COMPANY (US) 1988-05-03 US disclosed
US-4740233-A Substituted 1,2,4-triazolo[1,5-a]-pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1988-04-26 US disclosed
EP-0142152-A2 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1985-05-22 EP disclosed