SCHEMBL9832798

SCHEMBL9832798

CCOC(=O)c1cccc(Cl)c1NS(=O)(=O)c1nc2nccc(C)n2n1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.54
L3MBTL1 Q9Y468 1/20 0.44
MAPK1 P28482 4/20 0.43
POLB P06746 4/20 0.43
KMT2A Q03164 3/20 0.43
TSHR P16473 1/20 0.43
MAPT P10636 3/20 0.42
HTT P42858 2/20 0.42
LMNA P02545 4/20 0.41
KDM4E B2RXH2 3/20 0.41
GAA P10253 2/20 0.41
NPC1 O15118 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
MEN1 O00255 2/20 0.41
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9832974 0.91 ALDH1A1 (0.43) ALDH1A1L3MBTL1MAPK1POLBKMT2A
SCHEMBL9831492 0.90 ALDH1A1 (0.56) ALDH1A1L3MBTL1MAPK1POLBKMT2A
SCHEMBL9832897 0.89 ALDH1A1 (0.49) ALDH1A1L3MBTL1MAPK1POLBKMT2A
SCHEMBL9831723 0.89 ALDH1A1 (0.54) ALDH1A1L3MBTL1MAPK1POLBKMT2A
SCHEMBL9832261 0.89 ALDH1A1 (0.49) ALDH1A1L3MBTL1MAPK1POLBKMT2A
SCHEMBL9832070 0.88 L3MBTL1 (0.41) ALDH1A1L3MBTL1MAPK1POLBKMT2A
SCHEMBL9832778 0.88 ALDH1A1 (0.54) ALDH1A1L3MBTL1POLBKMT2ATSHR
SCHEMBL9833575 0.87 ACLY (0.43) ALDH1A1L3MBTL1MAPK1POLBTSHR
SCHEMBL9833484 0.86 ALDH1A1 (0.52) ALDH1A1L3MBTL1MAPK1POLBKMT2A
SCHEMBL10659813 0.86 MAPT (0.41) ALDH1A1MAPK1KMT2ATSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0142152-B1 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1991-03-20 EP claimed
EP-0142152-A2 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1985-05-22 EP claimed
EP-0142152-B1 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1991-03-20 EP disclosed
EP-0330137-A1 Intermediate compounds for the preparation of 1,2,4-triazolo [1,5-a]pyrimidine-2-sulfonamides DowElanco (US) 1989-08-30 EP disclosed
US-4755212-A Novel substituted 1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonamides and compositions and method for inhibiting pollen formation in corn THE DOW CHEMICAL COMPANY (US) 1988-07-05 US disclosed
US-4741764-A SUPPRESSION OF NITRIFICATION OF AMMONIUM NITROGEN IN THE SOIL THE DOW CHEMICAL COMPANY (US) 1988-05-03 US disclosed
US-4740233-A Substituted 1,2,4-triazolo[1,5-a]-pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1988-04-26 US disclosed
EP-0142152-A2 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1985-05-22 EP disclosed